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8-{[3-(cyclopentyloxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2R,3S,6R)-3-(4-fluorophenyl)-5-[(2-methoxypyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(4S,4aS,8aS)-1-(2-hydroxypyridine-3-carbonyl)-4-phenyl-decahydroquinolin-4-ol
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-one
1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-N-(pyridin-4-ylmethyl)piperidin-4-amine
N4,N4,5-trimethyl-N2-[3-(pyridin-4-yl)propyl]pyrimidine-2,4-diamine
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-[2-(cyclohexylmethyl)morpholin-4-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(4-methylbenzoyl)pyrrolidin-3-yl]methanol
4-(7-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)morpholine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2,2-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]oxane-4-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2-{2-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
6-(aminomethyl)-N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N,2-dimethylpyrimidin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methoxypyrazin-2-yl)piperidin-3-ol
N-(2-methoxypyridin-3-yl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzamide
1-methyl-6-(propan-2-yl)-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-1H-pyrazolo[3,4-d]pyrimidine
9-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(2,5-dihydro-1H-pyrrole-2-carbonyl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(2-methoxynaphthalen-1-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylsulfanyl)propan-1-one
7-[(4-fluorophenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
{2-[2-methyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]-2-oxoethyl}urea
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-N-methylpyridin-2-amine
N-(2-{7-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
1-[1'-(quinolin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
4-phenyl-3-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-hydroxy-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
1,3-dimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-methyl-2-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-N-methylpiperidine-2-carboxamide
3-[3-(5-methylfuran-2-yl)-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
5-(piperidine-1-carbonyl)-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
1-(4-methylphenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
N-(3-chloro-4-methylphenyl)-3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidine-1-carboxamide
(4aR,8aS)-1-(1-methyl-1H-pyrazole-5-carbonyl)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine
(2R,3R)-1'-(4-amino-5-methylpyrimidin-2-yl)-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]propanamide
4-[4-(morpholin-4-yl)benzoyl]-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-dimethyl-3-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]aniline
3-cyano-N-propyl-N-(pyridin-3-ylmethyl)benzamide
(1R,7S)-3-cycloheptyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]benzonitrile