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methyl 1-{[1-(cyclohexylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperidine-4-carboxylate
(3aS,6aS)-2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-3-cyclobutyl-4-methyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)pyrrolidin-3-ol
1-(2-{1-[2-(2,3,6-trimethylphenoxy)acetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
3-(azocane-1-carbonyl)-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
(1S,5R)-3-benzoyl-6-(1-methylcyclopropanecarbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}piperidin-3-yl)methanol
6-[methyl(2-methylpropyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
2-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-{[(2-hydroxyethyl)(methyl)amino]methyl}-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]benzamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}pyrimidin-2-amine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
(3R,4R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(hydroxymethyl)piperidin-3-ol
9-(5-fluoro-2-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}quinolin-4-ol
N-(3-methoxyphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
1-methyl-3-(4-{4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]piperidin-1-yl}phenyl)imidazolidin-2-one
2-[(2-cyclohexylpyrimidin-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(2-phenylethyl)piperidine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-methylpyrimidin-2-amine
2-{9-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-{3-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
3-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}-2-(thiophen-2-ylmethyl)propan-1-ol
6-(benzyloxy)-4-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
7-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[4-(pyridin-2-yl)pyrimidin-2-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-methoxy-1-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(pyridin-3-ylmethyl)piperazine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
[(4aS,8aR)-6-(3-fluorobenzoyl)-1-(1H-imidazol-4-ylmethyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
3-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}benzonitrile
2-[2-(1H-imidazol-1-yl)ethyl]-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
N-[(2,3-dimethoxyphenyl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
{1-methyl-4-[(4-phenylphenyl)methyl]piperazin-2-yl}methanol
4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)azepan-3-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(piperidin-1-ylmethyl)benzamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]oxane-4-carboxamide
(2R,6R)-4-[3-(pyridin-3-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide