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methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3,5-dimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-oxazole-4-sulfonamide
3-(2-chloro-4-fluorophenyl)-4-methylbenzamide
6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine-2,4-diamine
8-(cyclopentylcarbamoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
N-(3-ethylphenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(3S,4S)-1-(cyclopentylcarbamoyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-(2-methoxyethyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
1-cyclohexanecarbonyl-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-methyl-3-(1H-pyrazol-4-yl)-N-[1-(thiophen-2-yl)ethyl]propanamide
3-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-[4-chloro-3-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
N-[1-(4-methanesulfonylphenyl)propyl]-2-[methyl(piperidin-4-yl)amino]acetamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2-hydroxy-6-methylpyridine-3-carbonyl)piperidin-3-yl]propan-1-one
1-[(3-fluorophenyl)methyl]-4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
4-(piperidin-1-ylmethyl)-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
3-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}benzoic acid
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 5-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(3-benzoylpiperidin-1-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[4-(1-benzofuran-2-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-3-ol
1-(2-benzyl-1,3-thiazole-4-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
1-(2-fluorophenyl)-4-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]piperazine
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)propan-1-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(naphthalen-1-yl)acetamide
3-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(1-ethyl-1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine
2-phenyl-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3R)-1-{2-[(thiophen-2-ylmethyl)amino]benzoyl}pyrrolidin-3-ol
4-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}benzene-1-sulfonamide
1-[4-({[2-(furan-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(3R,4S)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-propylpyrrolidin-3-amine
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(2-chlorophenyl)methyl]-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]methylamine
N,N-dimethyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-N-(2-acetamidoethyl)-3-phenylpropanamide
3-(3-methyl-1H-pyrazol-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-(diethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
1-(4-chlorophenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)cyclobutane-1-carboxamide
8-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-(2-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid