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1-(cyclobutylmethyl)-3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
5-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)quinoline-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(5-chloro-2-methoxypyridin-4-yl)-N,N-dimethylbenzamide
N-(4-{4-[(1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)-3-phenylpropanamide
N-[(3,4-dimethylphenyl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
1-[1'-(3,6-dimethylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
6-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]-1,2,3,4-tetrahydronaphthalen-1-one
N,4-dimethyl-5-[3-(3-methylphenyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(trifluoromethyl)pyrimidine
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-cyclopentyl-5-methyl-1H-pyrazole-4-carboxamide
(1R,5R)-6-benzyl-N-[(2-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(1-{6-[(oxolan-3-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
3-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-ethyl-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridine-3-carboxamide
2-amino-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4-methylpyrimidine-5-carboxamide
(3aR,6aR)-2-(3-fluoro-2-methylbenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-ethylpiperazin-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
3-{[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]amino}-2,2-dimethylpropan-1-ol
3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
(2S,4R)-N-ethyl-4-(4-{[(2E)-3-phenylprop-2-enamido]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-carbamoyl-4-ethoxyphenyl)-5-methyl-1H-pyrazole-3-carboxylic acid
3-fluoro-2-methoxy-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]benzamide
2-[5-(3-acetylphenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
methyl (2S,4S)-4-(2,3-dihydro-1,4-benzodioxine-5-amido)-1-methylpyrrolidine-2-carboxylate
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(methylsulfanyl)propyl]propanamide
{1-[2-(2-chloro-5-methylphenoxy)ethyl]piperidin-4-yl}(pyridin-3-yl)methanol
N-benzyl-1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-methylpiperidine-3-carboxamide
4-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}thiomorpholine
(1R,5S)-8-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
1-(3-cyclopentylpropyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
9-(2-phenoxyethanesulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-methyl-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}thiophene-2-carboxamide
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
5-({cyclopropyl[(4-ethoxyphenyl)methyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-1,2,3-triazole
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4,4-difluoropiperidine
1-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
2-(methoxymethyl)-6-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[5-(4-cyclohexylpiperazine-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
5-cycloheptyl-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine