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2,2-dimethyl-1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
4-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]benzonitrile
2-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
2-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methoxy}-N-ethylbenzamide
(2S,4R)-4-amino-1-[2-(1-benzylpiperidin-4-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
(3S,4R)-1-(3-fluoro-4-methylbenzenesulfonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-ethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}acetamide
1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
3-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-ol
(1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyridine
3-[(4S)-2,5-dioxoimidazolidin-4-yl]-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]propanamide
1-{2-methoxy-6-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
(1S,5R)-1,3,3-trimethyl-6-[1-(propan-2-yl)-1H-pyrazole-3-carbonyl]-6-azabicyclo[3.2.1]octane
3-[(benzylsulfamoyl)(propan-2-yl)amino]propanamide
N-(1H-imidazol-2-ylmethyl)-5-[1-(2-phenylethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-(2-methylpropyl)-N-[2-(morpholin-4-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopentyl-1-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-8-fluoroquinoline-2-carboxamide
5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-({5-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]furan-2-yl}methyl)-N-methylmethanesulfonamide
3-[(2R,3R,6R)-5-[(2-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1,2,3,4-tetrahydroisoquinoline
3-(3-fluorophenoxymethyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
2-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]-1,3-thiazole-4-carboxamide
3,4,7-trimethyl-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
N-{3-[6-amino-5-cyano-4-(3-methylthiophen-2-yl)pyridin-2-yl]phenyl}acetamide
6-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1,4-dimethyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-indole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-(4-methyl-1,4-diazepan-1-yl)acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(3-propoxypropyl)pyrimidin-2-amine
N-[4-(dimethyl-1,2-oxazol-4-yl)-2-methylphenyl]pyridine-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-(2-chlorophenyl)-2-hydroxy-1-{4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-[3-(benzyloxy)propyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-{[benzyl(methyl)amino]methyl}-3-(1-phenylcyclopropaneamido)thieno[2,3-b]pyridine-2-carboxylate
2-chloro-6-methoxy-4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(thiolan-3-yl)-1,4-diazepan-2-one
(1S,4S)-5-methanesulfonyl-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-methylphenoxy)acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(4-hydroxy-3-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(thiophen-3-yl)acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
N-(1-hydroxybutan-2-yl)-2-oxo-N-(thiophen-2-ylmethyl)-2H-chromene-3-carboxamide
(1R,7S)-3-(2-ethoxyethyl)-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-3-(pyridin-4-yl)propanamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine