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N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-4-methoxybenzamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]pyridine-3-carboxamide
2-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-7-methyl-2,7-diazaspiro[4.4]nonane
4-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)thiomorpholine
3-amino-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-N-propyl-3-(pyridin-4-yl)propanamide
(1R,3S)-7-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-[4-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)phenyl]ethan-1-one
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[(5-methylpyrazin-2-yl)methyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{[(3S,4R)-4-ethoxyoxolan-3-yl]amino}-N-[(2-fluorophenyl)methyl]acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)acetamide
2-[(3-methoxyphenyl)amino]-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]butanamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(2R,6S)-2,6-dimethyl-4-[2-(morpholine-4-carbonyl)-2,3-dihydro-1H-inden-2-yl]morpholine
2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
9-(3-methoxy-5-methylthiophene-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1S,5R)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[(4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}benzonitrile
(3S,9aR)-3-(cyclohexylmethyl)-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
diethyl({3-[4-(pyridin-3-yl)piperazine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-{[1-(oxan-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
methyl 2-[(4aS,8aR)-decahydroisoquinoline-2-sulfonyl]-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclopentyl-4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
(3R,4R)-3-cyclopropyl-4-methyl-1-{2-[(2-phenylethyl)sulfanyl]pyridine-3-carbonyl}pyrrolidin-3-ol
(3S,4S)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
2-{pyrazolo[1,5-a]pyridin-7-yl}-3-(pyrrolidin-1-yl)pyrazine
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]azepan-4-amine
N-(1H-pyrazol-3-yl)-5-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-hydroxy-2,2-dimethylpropyl)-5-methoxybenzamide
N-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]-N-methylacetamide
1-(azepan-1-yl)-3-(3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
4-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-methoxypyridine-3-carbonitrile
N-(1-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-methoxybenzamide
7-[(3,4-difluorophenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-carbamoyl-2-methylphenyl)azocane-1-carboxamide
N-methyl-N-[(5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}furan-2-yl)methyl]methanesulfonamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(1,4-dioxan-2-ylmethyl)-5,6-dihydrophenanthridin-6-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(3-hydroxyadamantan-1-yl)ethyl]propanamide
N,1-dimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5,6-dimethylpyrimidine
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(3R,5S)-N,1-bis(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide