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5-(2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4S)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-(naphthalen-2-yl)piperidin-3-ol
(3aR,6aR)-2-[2-(4-chlorophenyl)acetyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-benzyl-1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidin-4-ol
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-1-phenylmethanesulfonamide
benzyl 3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopiperidin-1-yl)propanamide
2-[2-(propan-2-yloxy)phenyl]-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
5-(2,6-dimethoxyphenyl)-2-(trifluoromethyl)pyridine
(3R,4R)-1-cyclohexanecarbonyl-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-(methylsulfanyl)-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
5-(4-fluorophenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
9-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,9-diazaspiro[5.6]dodecane
N-[(1-hydroxycyclohexyl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[4-(3,5-dichloro-4-methylbenzoyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(5-methylthiophen-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-ethyl-8-(furan-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-5-(7-fluoro-4-methylquinolin-2-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-chloro-5-sulfamoylphenyl)-4-(2-methoxyethyl)piperazine-1-carboxamide
2-[(3-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}phenyl)amino]acetic acid
3-{5-[(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
3-[5-(6-aminopyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(2-chloro-4-fluorophenoxymethyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-(1-{1-[2-(azepan-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
2-(ethylamino)-N-(2-oxoazepan-3-yl)pyrimidine-5-carboxamide
1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carbonitrile
5-methoxy-2-[2-(3-phenylpropyl)morpholine-4-carbonyl]phenol
4-(1-methylpiperidin-4-yl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
9-(3-methoxybenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(aminomethyl)-2-[(2,6-dichlorophenyl)methyl]-3,4-dihydropyrimidin-4-one
(3aR,7aS)-2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-ethyl-4-{[2-(2-phenyl-1,3-thiazol-5-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
2-[1-(thiophen-2-ylmethyl)-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
4-(1-ethyl-1H-imidazol-2-yl)-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2-methylphenyl)(pyridin-4-yl)methyl]acetamide
2-[2-(1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethyl]pyridine
methyl (2S,4R)-4-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzamido]-1-methylpyrrolidine-2-carboxylate
N-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N,N-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7,7-dimethyl-2-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[3-(methylsulfanyl)phenyl]acetamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
4-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
4-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol