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(1S,5R)-3-[2-(2-ethylphenoxy)ethyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
3-{2-oxo-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2,5,6-tetramethylpyrimidin-4-amine
(4aR,7aS)-1-ethyl-4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-methoxy-1-{4-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
7-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,3-diazepane-2,4-dione
4-{1-[(3-methoxyphenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}pyridine
N-[(1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
2-cyclopropyl-5-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
2-(3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-5-methyl-1H-pyrazol-1-yl)-N-methylacetamide
3-(pyridin-4-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(naphthalen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-[3-(2-methoxyphenyl)phenyl]-3-[1-(pyrrolidin-1-yl)propan-2-yl]urea
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-ethyl-5-methylpyrimidin-2-amine
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
3-(azepane-1-carbonyl)-5-(4-benzylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-ethyl-N-methylpyrimidin-4-amine
3-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-fluoro-2-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)quinolin-4-ol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,3-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(4-acetylpiperazin-1-yl)-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropan-1-one
(3S,9aR)-8-(4-ethylbenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(ethylsulfanyl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
2-methyl-6-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
(2R)-2-amino-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenylethan-1-one
3-(3-fluorophenyl)-4-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanoyl}piperazin-2-one
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,9aR)-8-(2-chlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[3-(1H-imidazol-1-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-(3-cyanophenyl)-4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
4-{[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]sulfonyl}-N-tert-butylbenzamide
4-benzyl-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine
(1S,6R)-9-(thian-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-N4-(propan-2-yl)pyrimidine-2,4-diamine
[2,4,6-trimethyl-3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)phenyl]methyl acetate
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
1-(naphthalen-1-ylmethyl)-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(4-fluoropiperidine-1-carbonyl)-5-methoxybenzoic acid
benzyl({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-5-(methoxymethyl)furan-2-carboxamide