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N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-5-chlorofuran-2-carboxamide
1-[(2,3-difluorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
5-(1-benzofuran-5-yl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
[(5-methylthiophen-2-yl)methyl]({[5-(oxan-2-yl)furan-2-yl]methyl})(pyridin-4-ylmethyl)amine
2-[3-(2-methylpropyl)-5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H-1,2,4-triazol-1-yl]pyridine
(4aS,8aR)-6-[3-(methylsulfanyl)propanoyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2,3-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinoxaline-6-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-amino-4-[4-(2-hydroxyethoxy)phenyl]-6-(1H-indol-3-yl)pyridine-3-carbonitrile
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}piperidine
4-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidine-3-carboxylic acid
3,3-dimethyl-1-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
5-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-methylurea
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3-thiadiazole-4-carboxamide
N-(4-fluorophenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}benzamide
N-[(3-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)methyl]propanamide
5-(2-phenyl-1H-imidazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
2-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[4-(trifluoromethyl)pyrimidin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
[(2-ethylpyrimidin-5-yl)methyl][(2-fluorophenyl)methyl]propylamine
7-(2,3-dimethyl-1H-indole-5-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
1-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(dimethylamino)ethyl]-3,3,3-trifluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)propanamide
8-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(3R,4R)-1-(2,3-difluoro-6-methoxybenzoyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-hydroxy-1-(3-phenylpropyl)-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}piperidin-2-one
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
N-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-benzyl-3-ethyl-1-(3-hydroxybenzoyl)-1,4-diazepan-5-one
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4S)-4-amino-N-ethyl-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)pyrrolidine-2-carboxamide
3-ethyl-8-(furan-3-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,4S)-4-hydroxy-1-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperidine-2-carboxylic acid
6-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butane-1-sulfonamide
2-cyclopropyl-9-(4,6-dimethylpyrimidin-2-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
1-ethyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-cyclopentyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-6-oxopiperidine-3-carboxamide
8-chloro-2-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}quinoline
5-{[4-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methylpiperazin-1-yl]sulfonyl}isoquinoline