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2-methyl-5-propyl-4-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
2-[3-(3,4-difluorophenyl)-5-(2-ethylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-phenoxypropan-1-one
N-(2-methylpropyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-({2-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(3aS,6aR)-N-cyclohexyl-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
3-(1-methanesulfonylpiperidin-4-yl)-1-[3-(1H-pyrazol-5-yl)phenyl]urea
(3R,4R)-1-[(2,3-difluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-[(2R)-2-hydroxypropanoyl]-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-(4-chlorophenyl)-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]butanamide
5-chloro-1,3-dimethyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazole-4-sulfonamide
4-(piperidin-3-yl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
4-({4-[1-propyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)morpholine
5,6-dimethyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-hydroxy-1-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(methylsulfanyl)butan-1-one
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
11-[benzyl(2-hydroxyethyl)amino]-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-methyl-N-[(1R,2S)-2-phenylcyclopropyl]-3-propyl-1H-pyrazole-5-carboxamide
3,5-dimethyl-1-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
2-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-methylpropanamide
1-{1-[(3E)-pent-3-enoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1S,6R)-9-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
3-(3,5-difluorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
2-amino-4-(3-fluoro-4-methylphenyl)-6-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1S,6R)-9-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-cyclohexyl-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-ethyl-2-(4-fluorophenoxy)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
6-ethyl-N,1,5-trimethyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
6,8-dimethyl-3-(2-methylcyclohexyl)-3,4-dihydroquinazolin-4-one
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
2-methoxy-1-{1'-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-(2,3-dimethylphenoxy)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-[2-(dimethylamino)ethyl]-1-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-3-(oxolan-2-ylmethyl)urea
1-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
{3-ethyl-1-[5-(pyrrolidin-1-yl)pyridazin-3-yl]piperidin-3-yl}methanol
methyl 3-(4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)propanoate
2-(2-methyl-1,3-thiazol-4-yl)-4-oxo-N-phenyl-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]-S-(thiophen-2-yl)ethane-1-sulfonamido
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}propanamide
1'-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
5-(2,4-dichlorophenyl)pyridin-3-amine
2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]acetic acid
N-(2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)acetamide
3-phenyl-1-{1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}propan-1-one