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N-(2-methylprop-2-en-1-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-1-methylpiperidin-4-amine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-ethylphenyl)methyl]piperidine
2-amino-2-methyl-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[4-(3-methoxyphenyl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
8-(cyclohex-3-en-1-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
(4aS,8aR)-1-propyl-6-(quinoxaline-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-[2-(1H-1,3-benzodiazol-2-yl)phenoxy]ethan-1-ol
(1-{[1-(quinoline-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-3-(hydroxymethyl)piperidin-3-ol
3-[4-fluoro-3-(hydroxymethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
2-amino-4-(4-fluoro-2-methylphenyl)-6-(pyridine-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[4-(4-benzyl-4-hydroxypiperidine-1-carbonyl)piperidin-1-yl]-2-methoxyethan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(2-ethyl-1H-imidazol-1-yl)propanamide
ethyl 1-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-benzylpiperidine-3-carboxylate
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
3-{[4-(9H-purin-6-yl)piperazin-1-yl]methyl}piperidin-3-ol
(2S,4R)-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
2-(cyclopentylmethyl)-N-(1-hydroxy-2-methylpropan-2-yl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
2-(3-chloro-2-fluorophenyl)benzamide
2-[3-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrazine
N-[(2-methylphenyl)methyl]-6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carboxamide
7-chloro-3-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]quinolin-4-ol
2-amino-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-methylpyrimidine-5-carboxamide
1-{3-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-3-propylpiperidine-3-carboxylic acid
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[3-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
5-[5-(2,3-dimethyl-1H-indol-5-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
6-(dimethylamino)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyridine-3-carboxamide
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
N-[(1-benzylpiperidin-4-yl)methyl]-1-tert-butyl-N-methyl-1H-pyrrole-3-carboxamide
3-{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}-2,2-dimethylpropan-1-ol
3-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
2-(2H-1,3-benzodioxol-5-yl)-6,7-dimethoxyquinazolin-4-amine
N,N-dimethyl-5-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)-1,3-thiazol-2-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,5,7-trimethylquinoline-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
(1S,5R)-6-benzyl-3-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{4-[1-(2-fluorophenyl)piperidin-4-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-benzyl-8-(1-methoxypropan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,3S)-3-methoxy-7-(5-methyl-2-phenylfuran-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine