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1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
4-methyl-1-({3-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidine-4-carbonitrile
2-(1H-imidazol-1-yl)-N-[(3-methoxyphenyl)methyl]acetamide
N-methyl-N-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)thian-4-amine
N-(1,4-dioxan-2-ylmethyl)-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
(1R,5S)-6-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
1-phenyl-N-[2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]cyclopropane-1-carboxamide
5-[4-(1H-imidazol-1-yl)phenoxy]-1-azabicyclo[3.2.1]octane
N-methyl-N-[2-(morpholin-4-yl)propyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}methanol
1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
8-chloro-2-(furan-2-yl)-N-[2-(1H-imidazol-1-yl)ethyl]quinoline-4-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(4-methylpyridin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(4-fluorophenyl)cyclopentyl]methyl}acetamide
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
N-butyl-N-[(4-chlorophenyl)methyl]-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-hydroxy-3-phenylpropan-1-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[4-(1H-pyrazol-1-yl)butanoyl]pyrrolidin-3-yl]acetamide
4-[2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)ethyl]morpholine
N-[(4-fluorophenyl)methyl]-3-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
4,4,4-trifluoro-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
1-methyl-5-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
4-amino-N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-2-carboxamide
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
(3aR,5R,6S,7aS)-5,6-dihydroxy-N-(4-methanesulfonylphenyl)-octahydro-1H-isoindole-2-carboxamide
N-(2-ethoxybutyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-methyl-1-(1-{6-[(oxan-4-yl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
(3R,4R)-4-(azepan-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
5-cyclopropyl-3-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
methyl({1-[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-4-ylmethyl)amine
2-[({[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-5-methoxyphenol
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-4-oxo-N-(oxolan-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(trifluoromethyl)benzamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
N-[(2R,3R)-1'-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N,N-bis(1,3-oxazol-4-ylmethyl)-4-(1H-pyrazol-4-yl)butanamide
6-cyclopentyl-1-methyl-N-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(4-chlorophenyl)-3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}propanamide
5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(2,2,2-trifluoroethyl)acetamide
(1S,3R)-3-amino-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]cyclopentane-1-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]propanamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
N-(6-methoxy-2-methylquinolin-4-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide