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N-ethyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-amido]piperidine-1-carboxamide
ethyl 4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-amido}piperidine-1-carboxylate
1-[3-(furan-2-yl)phenyl]-3-[1-(methoxymethyl)cyclopentyl]urea
(2S,4S)-N-ethyl-4-{4-[2-(thiophen-2-ylformamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]benzamide
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[4-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-(cyclooctylamino)-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-fluorophenyl)-N-({7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
N-[(3S,4R)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxyphenyl)methyl]piperidine
3-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-[(3-methoxyphenyl)methyl]propanamide
(3S,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-{[3-(pyridin-3-yloxy)propyl]amino}propan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}acetamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]pyrrolidine-2-carboxamide
2-(pyrimidin-5-yl)quinoline-4-carboxylic acid
(3aS,6aR)-2-oxo-N-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
1-(2-methoxyethyl)-N3-(3-methylbutyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
dimethyl(2-{4-[4-(methylsulfanyl)benzoyl]morpholin-2-yl}ethyl)amine
3,3-difluoro-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
3-[ethyl({[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-[(3,4-dimethoxyphenyl)methyl]-N-(1-hydroxypropan-2-yl)-1,3-benzoxazole-6-carboxamide
1-[(1-methylpiperidin-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
2-(1-benzyl-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
methyl 1-[(3R,5S)-1-(1-benzylpiperidin-4-yl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
2-{4-[3-(1-methoxyethyl)phenyl]-1H-pyrazol-1-yl}acetamide
4-benzyl-3-ethyl-1-(morpholine-4-carbonyl)-1,4-diazepan-5-one
methyl 2-(cyclohexylsulfamoyl)-6-(3,5-difluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-5-{[(1-phenylcyclohexyl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(hydroxymethyl)-N-(4-methoxy-3,5-dimethylphenyl)piperidine-1-carboxamide
(4aR,8aS)-6-(propan-2-yl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)propan-1-ol
ethyl 2-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-2-yl)acetate
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]furan-3-carboxamide
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(pyrimidin-4-yl)ethyl]benzamide
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-N-methylacetamide
3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
5-(2,5-dimethylphenoxymethyl)-N-[(2R)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide
6-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1,3-benzothiazole