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N-(3-methylphenyl)-3-{[1-(oxolane-2-carbonyl)piperidin-4-yl]amino}propanamide
4-{2-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
(1R,5R)-6-[(3,4-difluorophenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluorophenyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-[2-(2-fluoro-5-methylphenyl)phenyl]ethan-1-amine
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3-(3-methoxyphenyl)-1H-pyrazole
4-[4-(4-methoxybutyl)piperazin-1-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-tert-butyl-2-{[1-(morpholin-4-yl)propan-2-yl]amino}acetamide
4-[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)piperidin-3-yl]benzoic acid
5-ethyl-N,2,3-trimethyl-N-(pyrimidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
1-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propan-1-one
N-cyclooctyl-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{4-[5-(cyclohexylsulfanyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
ethyl 4-[1-(adamantan-2-yl)piperidin-3-yl]piperazine-1-carboxylate
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-4-methyl-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-[(4-methyl-1H-imidazol-5-yl)methyl]cyclopropanamine
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)pyrrolidine-3-carboxylic acid
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(trimethyl-1H-pyrazol-4-yl)benzamide
1-[2-(benzyloxy)acetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(3-phenylpropyl)-1,4-diazepane
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
1-[3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]pyrrolidin-2-one
3-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
4,6-dimethyl-1-{3-oxo-3-[2-(pyridin-3-yl)piperidin-1-yl]propyl}-1,2-dihydropyrimidin-2-one
N-(4-chlorophenyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
3-(2-phenylethyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(3-methoxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]{[3-({1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
8-fluoro-2-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
(3R,5R)-N-methyl-5-(morpholine-4-carbonyl)-N-[2-(phenylsulfanyl)ethyl]piperidine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
1,4,6-trimethyl-3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-dihydropyridin-2-one
2-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]acetic acid
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
4-[1-(2-fluorobenzenesulfonyl)piperidin-3-yl]benzoic acid
4-(isoquinolin-4-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
6-tert-butyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-2-oxo-2,3-dihydropyrimidine-4-carboxamide
(3R,4R)-4-amino-1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-ol
(3aR,7aS)-2-(3-phenyl-1H-pyrazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-phenoxypropanamide
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide