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1-ethyl-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
(1R,5R)-6-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N5-[(3-chlorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-phenylethan-1-one
2,6-dimethoxy-3-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyridine
1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
4-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]quinoxaline-2-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}propan-1-one
2-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(6-methylpyridazin-3-yl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-[3-methyl-5-(1-phenyl-1H-1,2,3-triazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,2,3,4-tetrahydroisoquinolin-5-ol
3-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzene-1-sulfonamide
N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
2-(3-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
(3R,4R)-1-(1-benzofuran-5-carbonyl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
(3R,4S)-4-cyclopropyl-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]pyrrolidin-3-amine
7-(3,6-dimethylpyrazin-2-yl)-4-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,4R)-1-(3-chloro-2-methylbenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-{1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}propanamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-phenoxyethyl)piperazine
1-{6-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
2-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethyl)pyridine
[5-(1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
4-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decane-2-carbonyl}-1λ6-thiane-1,1-dione
4-({2-[4-(piperidine-1-carbonyl)phenyl]phenyl}methyl)morpholine
4-[2-(4-propoxyphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(1R,5S,8R)-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[(2R,3R)-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-fluorobenzamide
(1S,6R)-9-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-[1-(pyridine-2-carbonyl)piperidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
4-(2-fluorophenoxy)-1-(4-methylpyrimidine-5-carbonyl)piperidine-4-carboxylic acid
3-(4-tert-butylbenzoyl)-1-(thian-4-yl)piperidine
4-[2-(pyrrolidin-1-yl)phenyl]-4H-1,2,4-triazole
[(4aS,8aR)-6-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
1-({4-methyl-5-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
(1R,2S,6R,7S)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
1-{2-[1-(5-fluoro-1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
6,7-dimethyl-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-2H-chromen-2-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-(2-phenylethoxy)benzamide
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate