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1-[4-(5-methyl-2-phenylfuran-3-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[1-(pyrimidin-4-yl)ethyl]benzamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(5-fluoro-2-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
ethyl 3-({1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)propanoate
3-(1H-imidazol-1-ylmethyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
ethyl 4-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
(1R,5R)-6-benzyl-3-(3-chloro-5-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1,4-dioxan-2-ylmethyl)-2-(2-methoxyphenyl)acetamide
1-[1-methyl-5-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
2-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(3-methylthiophene-2-sulfonamido)acetic acid
2-(2-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]azepan-4-amine
8-(4,6-dimethylpyrimidin-2-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{4-[1-(1,2-oxazol-5-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenoxy}pyrimidine
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-(pyrazin-2-ylmethyl)acetamide
2-[(3-methoxypiperidin-1-yl)methyl]-6,8-dimethylquinolin-4-ol
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
6,8-dimethyl-2-({[(2S)-pyrrolidin-2-ylmethyl]amino}methyl)quinolin-4-ol
1-[4-(4-methylphenoxy)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
5-[4-(ethoxycarbonyl)piperazin-1-yl]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-methyl-6-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
2-(2,3-dihydro-1H-indol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)pyridine-3-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-{1-[(3-methoxyphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
(3R,4R)-3-cyclopropyl-4-methyl-1-(thiophene-2-carbonyl)pyrrolidin-3-ol
1-[4-({8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}amino)piperidin-1-yl]ethan-1-one
1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-(4-{[2-(benzylamino)pyrimidin-5-yl]methyl}morpholin-3-yl)-1-(2,5-dihydro-1H-pyrrol-1-yl)ethan-1-one
3-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-fluoro-3,4-dihydroquinazolin-4-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-3-yl)propan-1-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
3-methyl-7-[2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-benzyl-3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(6-methylpyridin-2-yl)methyl]propanamide
2-methoxy-N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
(3-{[(2S,5R)-5-{[methyl(1-methylpiperidin-4-yl)amino]methyl}oxolan-2-yl]methyl}phenyl)methanol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(9H-purin-6-yl)pyrrolidin-3-yl]acetamide
2-acetamido-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide