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N-cycloheptyl-5-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-{3-[(4aS,7aR)-4-[(5-methylfuran-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-3-oxopropyl}acetamide
N-cyclopropyl-1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
[(4-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}phenyl)methyl]dimethylamine
4-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
5-fluoro-2-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1,3-dimethyl-1H-indole
4-methyl-7-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-2H-chromen-2-one
1-{3-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
5-[(2-ethylpyrimidin-4-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-2-one
3-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-(adamantan-2-ylmethyl)-6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methoxy-1,2-dimethyl-1H-indole-3-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-cyclopentyl-4-(4-{[3-(1H-indazol-1-yl)propyl]amino}piperidin-1-yl)benzamide
2-{1-cyclohexyl-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{2-[3-ethyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2-fluorobenzamide
5-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[4-(dimethylamino)azepan-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-(3,4-dimethoxyphenyl)-4-phenyl-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazole
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-4-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-hydroxyphenyl)methyl]piperidin-3-yl]propanoate
(3S,4R)-4-phenyl-1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-butyl-8-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-phenyl-3-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)propanamide
3-(5-tert-butyl-2-methoxyphenyl)-1-[3-(4-methylpiperazin-1-yl)butyl]urea
methyl 6-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}pyrazine-2-carboxylate
5-(2,5-dimethylfuran-3-carbonyl)-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
1-{5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-methylphenyl}imidazolidin-2-one
(2S,4S)-4-cyclobutaneamido-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
(1S,3R)-3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclohexan-1-amine
1-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
2-cyclopentyl-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)acetamide
2-[2-({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
ethyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}[(3-fluorophenyl)methyl]amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazine
2-{4-phenyl-1-[2-(pyridin-2-yl)ethyl]-1H-imidazol-5-yl}benzonitrile
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridine-3-sulfonyl)piperidin-3-ol
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-(2-hydroxyethyl)-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-3-carboxamide
(3S,5R)-N3-butyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-hydroxy-2-methylbenzamide
2-[1-cyclohexyl-4-({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)piperazin-2-yl]ethan-1-ol