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N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,1,3-benzoxadiazole-5-carboxamide
2-(3-fluoro-4-methylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-[(1R,3R)-3-aminocyclopentyl]-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(1,3-thiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethyl)benzamide
8-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
4-(1-{[3-(trifluoromethyl)phenyl]methyl}azetidin-3-yl)morpholine
4-[1-(1-methylpiperidin-4-yl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl]pyridine
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,4-triazole
(4S)-3,3,4-trimethyl-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperidin-4-ol
3-{5-[2-(propylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
3-(3-chlorobenzoyl)-1-(thiophene-2-sulfonyl)piperidine
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(2,6-dimethylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(2-{[(2-chlorophenyl)methyl]sulfanyl}-N-methylacetamido)-N-methylbutanamide
2-{2-[3-(dimethylamino)propyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
2-methoxy-1-{1'-[3-(methylsulfanyl)propyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-[2-({[2-chloro-5-(methylcarbamoyl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
N-cyclopentyl-2,2-dimethyl-N-[(4-methylphenyl)methyl]cyclopropane-1-carboxamide
N-(3-ethoxypropyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
4-[4-(2-ethylbutanoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenoxy}ethan-1-ol
N-[(3S,4R)-4-propyl-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidin-3-yl]acetamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(thiophen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-3-(2-oxopyrrolidin-1-yl)propanamide
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}(methyl)[2-(morpholin-4-yl)propyl]amine
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-[(3-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-oxopropyl)(methyl)amino]-1λ6-thiolane-1,1-dione
2-methyl-4-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
2-(cyclopent-2-en-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(2-ethoxy-5-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenyl)methanol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-methoxy-N-methylpyrimidin-4-amine
9-(4-methoxypyrimidin-2-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N,N-dimethylpiperazine-1-sulfonamide
(2S,4R)-1-benzyl-N-methyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-{4-[(2-methylpropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(pyridin-4-yl)propan-1-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-cyclopropanecarbonyl-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}piperidine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
ethyl 1-(3,3-dimethylbutanoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-(2-methoxyethyl)-8-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(pyridin-2-yl)piperidin-1-yl]acetamide
3-(carbamoylmethoxy)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)benzamide
5-methyl-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-1-benzofuran-2-carboxamide
2-(3,4-dichlorophenyl)-4-(2-ethylpyrimidine-5-carbonyl)morpholine
4-(5-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol