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3-hydroxy-S-{2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}butane-1-sulfonamido
2-(methylsulfanyl)-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}pyrimidine
N-[(4-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)methyl]-2-methylpropanamide
(2S)-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidine-2-carboxamide
N-(4-butanamido-3-methoxyphenyl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-(furan-3-ylmethyl)-5-[1-(oxan-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
5-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-3-carboxamide
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
methyl(2-phenylethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}quinoxaline
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(4-methoxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
5-(2,6-difluoro-3-methylphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-2-carboxamide
1-(azepan-1-yl)-3-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1R,3R)-3-aminocyclopentyl]-1-[(4-methoxyphenyl)amino]cyclohexane-1-carboxamide
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2,4-dichlorophenoxy)-N-methylacetamide
(3R,4R)-3-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(oxan-4-yl)piperidin-4-ol
3-ethyl-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
4-[2-(2-chlorophenyl)acetyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(diethylamino)-3-[4-({[2-(4-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
ethyl 4-{[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}piperidine-1-carboxylate
2-{4-phenyl-1-[2-(phenylamino)ethyl]-1H-imidazol-5-yl}benzoic acid
methyl 4-[4-(3-hydroxy-2-methylbenzoyl)piperazin-1-yl]benzoate
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
(3aR,7aS)-2-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-cyclopropyl-1-[1-(quinoxaline-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidine-3-carboxylate
N-ethyl-1-(methoxymethyl)-N-[1-(4-methoxyphenyl)propyl]cyclobutane-1-carboxamide
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidine
1-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]cyclohexan-1-ol
3-[2-amino-4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-6-methylpyrimidin-5-yl]propanoic acid
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-ethyl-3,8-bis[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-chloro-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-3-[(4-fluorophenyl)methyl]piperidin-3-yl)methanol
2-[2-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)-4-(pyrimidin-2-yl)phenoxy]acetic acid
N-(2-aminoethyl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
(2R,6R)-4-[2-(benzyloxy)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-acetamido-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pentanamide
N3-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperidine-1,3-dicarboxamide
2-(1H-pyrazole-3-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(2-phenylethyl)piperidine