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N-(dicyclopropylmethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1,5-dimethyl-4-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
3-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-(8-methylquinolin-5-yl)urea
N-[(1s,4s)-4-[4-(diethylcarbamoyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]pyridine-2-carboxamide
1-{1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidin-3-yl}pyrrolidin-2-one
4-(4-chloro-1-methyl-1H-indazol-3-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
3-(3-fluorophenyl)-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-2-one
3-{[1-(3-phenylphenyl)piperidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(5-chloropyridin-2-yl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazine
6-fluoro-3-(4-methanesulfonylpiperazine-1-carbonyl)quinolin-4-ol
7-(7-chloroquinolin-4-yl)-2-oxa-7-azaspiro[4.5]decane
1-({3-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)-4-(prop-2-en-1-yl)piperazine
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-(2-hydroxyethyl)-5-methyl-4-{[(3S)-2-oxoazepan-3-yl]amino}-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}pyrimidine-5-carboxylic acid
3-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}phenol
2,5-dimethyl-6-[2-(pyridin-3-yl)piperidine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N,N,7,8-tetramethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)oxane-2-carboxamide
ethyl 1-[(3-methoxyphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-{2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl}phenol
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methoxypropanamide
1-[1-cyclohexyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
5-(5-ethylfuran-2-yl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
2-[(1-benzothiophen-5-ylmethyl)amino]-N-(2-acetamidophenyl)acetamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[3-(pyridin-3-yloxy)propyl]piperidine-3-carboxamide
2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}-3-(4-fluorophenyl)propanoic acid
1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
N-{2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
2-{[5-(morpholin-4-ylmethyl)-1,2-oxazol-3-yl]formamido}acetamide
5-(3,4-dichlorophenyl)-1,2,3,4-tetrahydroisoquinoline
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-{4-[3-(aminomethyl)pyrrolidin-1-yl]-6-oxo-1,6-dihydropyridazin-1-yl}butyl benzoate
8-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
methyl 6-{[methyl(propan-2-yl)amino]methyl}-3-(2-phenoxyacetamido)thieno[2,3-b]pyridine-2-carboxylate
N,3-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(1-hydroxycyclohexyl)methyl]-1,2-oxazole-3-carboxamide
N-(2-methylphenyl)-3-oxo-3-(2-phenylmorpholin-4-yl)propanamide
2-(1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazol-4-yl)benzoic acid
3-ethyl-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(4,4-difluoropiperidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(1H-pyrazol-1-yl)pyrimidine
2-methyl-4-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-thiazole
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-({3-methyl-7-[3-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidine