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1-ethyl-3,5-dimethyl-4-({2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}methyl)-1H-pyrazole
methyl 2-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1,3-oxazole-4-carboxylate
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-(2-methylpropyl)benzamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-6-(propan-2-yl)pyrimidin-4-amine
4-ethyl-4-[({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)methyl]hexanenitrile
5-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N,N-dimethylpyridin-2-amine
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)carbamoyl]amino}-4-methyl-N-propylbenzamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidine-3-carboxylate
7-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-chloro-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-methylquinoline
5-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
(3R,4R)-4-amino-1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-ol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(6-cyanopyridine-3-amido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
(2-methoxyethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})(thiophen-2-ylmethyl)amine
3-(4-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-[(4-ethylphenyl)methyl]-6-(2-hydroxyethyl)-N-(2-methoxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-fluoro-2-{1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
(benzylsulfamoyl)({2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
N-methyl-N-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
4-[(3-methylphenyl)sulfanyl]-1-(oxane-4-carbonyl)piperidine
2-({[(3R,4R)-1-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(1,3-benzoxazol-2-ylmethyl)-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(3-phenylpropyl)-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
(1S,2S)-2-{4-[3-(4-methoxyphenyl)propyl]piperazin-1-yl}cyclohexan-1-ol
1-(cyclopropylmethyl)-5-[2-(2-methoxyphenyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(2,3-dihydro-1-benzofuran-7-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
3-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-6-phenylpyridazine
1-ethyl-N-methyl-N-(2-methylpropyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(2-methylphenyl)-4-(oxolan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-cyano-6-[4-(1-ethoxyethyl)phenyl]-2-methylpyridine-3-carboxylic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)-2-methyl-1H-1,3-benzodiazole-5-carboxamide
7-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-2,4-dimethylquinoline
(2R)-N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyloxolane-2-carboxamide
2-benzyl-8-(5-methylthiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(furan-2-ylmethyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carboxamide
8-(2-hydroxypyridine-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
1-(3-{2-[2-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}propyl)piperidine-4-carboxamide
(2S,4R)-1-methyl-N-(propan-2-yl)-4-(4-sulfamoylbenzamido)pyrrolidine-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methylacetamide
2-(4-fluoropiperidin-1-yl)-4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}-1-phenylcyclohexane-1-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(2E)-3-(furan-2-yl)prop-2-en-1-yl](oxolan-2-ylmethyl)amine
4-(2-amino-5,6-dimethylpyrimidin-4-yl)-1λ6-thiomorpholine-1,1-dione
N-[2-(4-fluorophenyl)ethyl]-2-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine