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(4aR,8aS)-6-[(2-fluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
4-[4-(piperidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]-1-(1H-pyrazole-4-carbonyl)piperidine
1-{1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-(1-benzylpiperidin-3-yl)-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(propan-2-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-[(3R,4S)-3-(3,4-dihydro-2H-1-benzopyran-6-amido)-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
2-(4-methoxy-3-methylphenyl)pyridine-4-carboxamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
6-(2-methoxypyridin-3-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
(3R,4S)-3,4-dimethyl-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
5-(4,4-difluoropiperidine-1-carbonyl)-N-ethylpyrimidin-2-amine
(1S,4R)-2-{2-[1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-2-azabicyclo[2.2.1]heptane
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(3R,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dimethylpiperidin-4-ol
2-{2-[3-(methoxymethyl)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
(4aR,8aS)-1-[2-(dimethylamino)ethyl]-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridazine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
2-(2,4-dichlorophenoxy)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
5-[(2,3-difluorophenyl)methyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3S)-1-benzyl-N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-amine
2-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
{3-[(2,4-difluorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl}methanol
2-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
4-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(quinolin-6-yl)benzamide
1-tert-butyl-5-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(1-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-[(2-methoxyphenyl)methyl]propanamide
1-[5-(methoxymethyl)furan-2-carbonyl]-3-(2-phenylethyl)piperidine
N-(5-carbamoyl-2-methylphenyl)-4-(2-methoxyethyl)piperazine-1-carboxamide
6-(1-{imidazo[1,2-a]pyridin-6-ylmethyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
3-cyclopropyl-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N,5,7-trimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
methyl 7-oxo-3-[2-(pyridin-4-ylsulfanyl)acetyl]-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-3-methyl-1,2-oxazole-5-carboxamide
8-chloro-2-{[(1,2-oxazol-3-ylmethyl)amino]methyl}quinolin-4-ol
[1-({1-[(4-fluorophenyl)methanesulfonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{4-[3-({[(2-methoxyquinolin-3-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
5-[(1S,2R)-2-[(prop-2-en-1-yl)carbamoyl]cyclohexanecarbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-methoxy-2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(pyrrolidin-1-yl)pyrazine
4-(dimethylsulfamoyl)-N-(2-phenylphenyl)piperazine-1-carboxamide
2-(4-methoxy-3-methylphenyl)-3-(piperidine-1-carbonyl)pyridine