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2,5-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]furan-3-carboxamide
({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-{4-[2-(thiophen-3-yl)ethyl]piperazin-1-yl}pyrimidine
(3aR,5R,6S,7aS)-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
6-ethyl-2-methyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]quinoline-4-carboxamide
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}acetamide
6-[(diethylamino)methyl]-N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({7-[4-(4-fluorophenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
3-[3-(1-methoxyethyl)phenyl]-6-(pyrrolidin-1-yl)pyridazine
4-{4-[(6-fluoroquinolin-2-yl)methyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[1-(thiophen-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-amino-7-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
3-{2-oxo-2-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
1-(2H-1,3-benzodioxol-5-yl)-3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]urea
5,6-dimethyl-2-{3-[(4-phenylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-[(3,4-difluorophenyl)methyl]-3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
3-[3-(2-methoxyphenyl)phenyl]propanamide
3-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-1,2-dihydroquinoxalin-2-one
3-(4-fluorophenyl)-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}propanoic acid
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
dimethyl({4-[1-(oxane-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
(1S,4S)-5-[1-(4-chlorophenyl)cyclopropanecarbonyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-benzyl-N3-(cyclopropylmethyl)-N5-ethyl-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
1-[(4aR,8aR)-4a-hydroxy-7-[2-(2-methoxyphenoxy)ethyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-methyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
(4aR,7aS)-1-benzyl-4-(2-methylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-fluorophenyl)-N-(2-methoxyethyl)-2,2-dimethyl-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
4-{[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
N,N-dimethyl-5-{1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-imidazol-2-yl}pyridin-2-amine
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-dimethoxyphenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(2-methoxyphenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-2,8-dimethylquinoline
6-methoxy-N,1-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-indole-2-carboxamide
6-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
2-(diethylamino)-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopropanesulfonamide
4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-imidazole-2-carboxamide
2-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}-N-ethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-ethyl-5-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyridazine-4-carboxamide
(4aS,8aR)-6-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-{4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
5,7-dimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyrido[2,3-d]pyrimidin-4-amine
3-methoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
N-cyclopropyl-N-(1-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
1'-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}spiro[indene-1,4'-piperidine]