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3-methyl-1-(2-methylpropyl)-5-(oxolan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
8-[5-(3-cyclopropyl-1H-pyrazol-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]quinoline
1-tert-butyl-4-(6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-2-one
(3S,4R)-4-(hydroxymethyl)-1-{[4-(morpholine-4-sulfonyl)phenyl]methyl}piperidin-3-ol
1-({1-[6-(3-hydroxyphenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[1-(2-phenylethyl)piperidin-3-yl]pent-4-enamide
2-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methylphenyl)piperazine
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amine
(1S,5R)-3-benzyl-6-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
[(3R,4R)-1-(9H-fluoren-2-ylmethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-(dimethylamino)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
4-{[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
ethyl 4-[(4-methoxyphenyl)methyl]-1-(5-methylthiophene-2-carbonyl)piperidine-4-carboxylate
methyl 2-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}-1,3-oxazole-4-carboxylate
1-methyl-6-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-1-[3-(dimethylamino)pyrrolidin-1-yl]propan-1-one
6-[1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-{4-cyclohexyl-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-amino-4-(furan-2-yl)-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-({[2-(2-methyl-1H-indol-1-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-4-propylpyrimidine-5-carboxamide
6-(3-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
2-({[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-[(3-fluorophenyl)methyl]-4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperazine
N-[(2-methoxyphenyl)methyl]-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]acetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]propan-1-one
3-(pyrazin-2-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
2-{[5-(4-cyanophenyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
1-(3-methylfuran-2-carbonyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-4-[(3-methylphenyl)sulfanyl]piperidine
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}piperidin-2-one
3-[1-(4-fluorobenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(4-fluorophenyl)propyl]-5-methoxybenzamide
[(5-methylthiophen-2-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
3-({4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}methyl)-6-methyl-1,2-dihydroquinolin-2-one
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
3-[(4-fluorophenyl)formamido]-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(pyrrolidin-1-yl)pyridine
1-{[5-(benzenesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-3-ol
6-(2,5-dimethylfuran-3-yl)-N-(1-hydroxypropan-2-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(cyclopropylmethyl)-4-[(2-methylphenyl)methyl]-1,4-diazepane-6-carboxylic acid