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4-(2-hydroxyethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
methyl 1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperidine-2-carboxylate
N-{[1-(ethoxymethyl)cyclopropyl]methyl}-2,5,6-trimethylpyrimidin-4-amine
2-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-6-yl)acetic acid
N-methyl-4-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
2-(2,5-dimethylphenoxy)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
1-tert-butyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-methyl-1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)pentane-1,2-dione
3-ethyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-5-carboxamide
9-{[3-(2-aminoethyl)phenyl]methyl}-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidine-3-carbonyl}pyridine
4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-(1-propylcyclopropyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(adamantan-1-yl)-4-hydroxy-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylpyrimidine-5-carboxamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
8-[4-(difluoromethoxy)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-4-phenyl-1,4-diazepane
N-[3-(4-amino-5-methylpyrimidin-2-yl)phenyl]acetamide
3-(2-hydroxyphenyl)-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1H-pyrazole-5-carboxamide
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
3-cyclohexyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
4-{4-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N'-cyclopentyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]butanediamide
2-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-yl}oxy)pyrimidine
4-benzyl-3-ethyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,4-diazepan-5-one
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
(3S,4R)-4-phenyl-1-(2-propoxyacetyl)pyrrolidine-3-carboxylic acid
3-{[(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
1-[2-(4-chloro-1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-amino-4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
N,1-dimethyl-5-phenyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrrole-2-carboxamide
3-[(3R,4S)-1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
methyl[(1-{[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
1-(1-methylcyclohexanecarbonyl)-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
8-(1H-1,3-benzodiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
2-[2-chloro-4-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)phenoxy]acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
5-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
7-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
(1S,5R)-6-(3-methoxybenzoyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(2-fluorophenyl)methyl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzoxazole-6-carboxamide
(4aR,8aS)-6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-[2-(3-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-[(2-methylphenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
1-[2-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)pyrimidin-4-yl]piperidin-4-ol
4-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-oxazepane
(3S,4S)-1-[4-(cyclopropylcarbamoyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid