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1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
6-(4-methylpiperazin-1-yl)-1-(3-phenylpropyl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
2-(2-phenoxyethanesulfonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 4-{2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
N-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methanesulfonamide
1-(2-{2-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-2,3-dihydro-1H-indole
2-methyl-3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(3S,5R)-1-propanoyl-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1-(4-methylphenyl)piperazin-2-one
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanamide
2-hydroxy-4-(methylsulfanyl)-N-[2-(5-methylthiophen-2-yl)ethyl]butanamide
2-oxo-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
4-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}benzamide
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[3-(cyclopentyloxy)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
2-(1-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3-(2-hydroxyphenyl)-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-2-(4-ethylpiperazin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(2S)-2-{1-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}pyrrolidine-1-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-phenylpyrimidin-4-ol
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5-(propan-2-yl)pyrimidine
3-{[(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
6-(4-acetylphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
2-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-oxo-N-(propan-2-yl)acetamide
3-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4-methyl-2-(propan-2-yl)pyrimidine
(3R,9aR)-8-benzyl-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-oxazole-5-carboxamide
3-methoxy-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-(prop-2-ene-1-sulfonyl)piperidine-4-carboxylate
2-(2,3-dihydro-1H-inden-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
{3-[(3-methoxyphenyl)methyl]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl}methanol
1-[3-(dimethylamino)pyrrolidin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
3-[(1H-1,3-benzodiazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]propan-1-ol
N-[(3-hydroxypyrrolidin-3-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-phenylpyrimidin-2-amine
1-[(4aR,8aS)-6-(3-phenylpropyl)-decahydro-1,6-naphthyridin-1-yl]propan-1-one
N-(3-hydroxypropyl)-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
1-(3,4-difluorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-{[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]amino}propane-1,3-diol
(3S,4S)-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(piperidin-1-yl)pyrrolidin-3-ol
2-benzyl-9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(N-methyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)acetamide