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4-benzyl-1-(2-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2-oxoethyl)pyrrolidin-2-one
3-[3-(cyclopropylmethyl)-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
8-methyl-3-[2-(3-phenylpiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
(4aR,8aR)-7-[(5-acetylthiophen-3-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
5-chloro-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
5-(4-fluorophenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(3-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
3-cyclopropyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-{4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]morpholin-2-yl}ethan-1-amine
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methylphenol
2-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[3-(4-methylpiperazine-1-carbonyl)phenyl]-1-(pyridin-2-ylmethyl)urea
N-[(5-methylfuran-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N4-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-6-methylpyrimidine-2,4-diamine
2-methoxy-1-(4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-8-fluoroquinoline-2-carboxamide
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
2-[2-(5-methylfuran-2-yl)propyl]-1H-1,3-benzodiazole-5-carbonitrile
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-methyl-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-thiazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-ethyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-phenoxy-1-[3-(pyridin-4-yl)azetidin-1-yl]propan-1-one
2-{1-[(3-methoxyphenyl)methyl]-4-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
(1S,5R)-6-(2-methoxyethyl)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-fluoro-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-6-methylpyridine-3-carbonitrile
N-[2-(2,4-difluorophenyl)-1-(1-propanoylpiperidin-4-yl)ethyl]-N-methylcyclopropanecarboxamide
(2S,4S)-4-amino-N-(3-methoxypropyl)-1-methyl-N-[(4-methylphenyl)methyl]pyrrolidine-2-carboxamide
ethyl N-{3-[2-(thiophen-3-yl)-1H-imidazol-1-yl]phenyl}carbamate
2-chloro-9-methyl-3-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H-pyrido[1,2-a]pyrimidin-4-one
3-(dimethylamino)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]pyrrolidine-1-carboxamide
(3aS,6aR)-N-ethyl-3-[2-(4-fluorophenyl)ethyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
4-{[6-(4-methoxy-2-methylphenyl)pyridin-3-yl]methyl}morpholine
1-tert-butyl-N-[3-(4-methoxyphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
ethyl 5-{[3-(cyclohexylsulfanyl)propyl]carbamoyl}-1H-imidazole-4-carboxylate
1-{[1-(azepane-1-sulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N,5,7-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2,4-dimethoxybenzamide
1-(4-fluorophenyl)-4-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butane-1,4-dione
8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-fluoro-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[(2-methoxyphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide