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2-(methoxymethyl)-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-3-(1H-pyrazol-1-yl)benzamide
(3aS,6aS)-2-[(2,3-dichlorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(3-ethoxypropyl)amino]methyl}-6-methylquinolin-4-ol
4-methyl-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}benzamide
4-(4-methanesulfonylphenyl)-1H-indole
4-{1-azabicyclo[2.2.2]octan-3-yl}-N-(2-chloro-4-fluoro-5-methylphenyl)piperazine-1-carboxamide
N-benzyl-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-(2-ethyl-2,5-dihydroxypentyl)-2-methyl-1,3-thiazole-4-carboxamide
1-(2-chloro-5-sulfamoylphenyl)-3-[2-(2-hydroxyethoxy)ethyl]urea
3-(1-{2-[(2,6-dimethylphenyl)amino]propanoyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 2-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}acetate
4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridin-2-amine
3-(5-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(1S,9R)-11-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-[3-(2-phenylethyl)piperidin-1-yl]-6-(piperidine-1-carbonyl)pyrazine
(propan-2-yl)({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-[2-(3-chlorophenyl)ethyl]-4-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
1-{1'-[(2,2-dimethyloxan-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(2S,4R)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1S,5R)-6-benzyl-3-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(2-cyclopropylpyrimidine-5-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 5-(2,6-dimethoxypyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
methyl (2S)-1-{2-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
1-[4-(morpholine-4-carbonyl)phenyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
2-[1-(1-benzofuran-2-sulfonyl)azetidin-3-yl]pyridine
4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-(4-chloro-3-fluorophenyl)-4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
4-{2,9-diazaspiro[5.5]undecan-2-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
N-(2-methoxyethyl)-2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-cyclopropanecarbonyl-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,N-dimethyl-2-[methyl({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amino]propanamide
4-[3-oxo-4-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepane-1-carbonyl]pyridin-1-ium-1-olate
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(6-methoxypyrimidin-4-yl)-4-(pyridin-2-yl)piperidin-4-ol
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxylate
2-oxo-2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
1-cyclopentyl-4-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
5-ethyl-N4-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]pyrimidine-2,4-diamine
7-(1,3-thiazol-2-yl)-N4-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(pyrimidin-2-yl)piperidin-4-amine
3-(cyclopropylmethyl)-1-(6-methylpyridazin-3-yl)piperidine-3-carboxylic acid
1-(2-methoxyphenyl)-3-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
2-(2-methoxyethyl)-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-methylpyridine-3-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[2-(2,4-dimethoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
12-(4-ethylpiperazine-1-carbonyl)-15-methyl-9-(3-methylthiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one