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(3S,4R)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-methylpiperidine-3,4-diol
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
1-[3-(benzyloxy)phenyl]-3-{[4-(hydroxymethyl)oxan-4-yl]methyl}urea
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}phenyl)-3-methoxypyrrolidine-1-carboxamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methoxybenzamide
2-(hydroxymethyl)-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-1H-1,3-benzodiazole-5-carboxamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
(1R,5R)-6-{imidazo[1,2-a]pyridine-2-carbonyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-2-[(dimethylamino)methyl]phenol
5-methyl-2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,3-benzoxazole
5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
ethyl 3-benzyl-1-(thiophene-3-sulfonyl)piperidine-3-carboxylate
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methoxyfuran-2-carboxamide
3-cyclopropyl-1-(3,4-difluorophenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-phenoxyethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-(2-methoxyacetyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
1-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)cyclohexane-1-carboxamide
2-methanesulfonamido-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
2-(dimethylamino)-4-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrimidine-5-carboxamide
2-[4-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]benzonitrile
4-(1H-1,3-benzodiazol-1-yl)-1-[(1-methyl-1H-indol-2-yl)methyl]piperidine-4-carboxylic acid
N-benzyl-N-[(1R,3S,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]-5-propyl-1,2-oxazole-3-carboxamide
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-3-propyl-1H-pyrazole-5-carboxamide
6-methyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,6R,8aS)-2-(4,6-dimethylpyrimidin-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-phenoxypropan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidine-2-carboxamide
1-(furan-2-ylmethyl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
1-methyl-4-{1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
ethyl 1-(3-phenylpropyl)-5-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-({[(3R,4R)-1-(4-fluoro-3-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
4-(2-methoxyacetyl)-N-[2-(5-methylfuran-2-yl)phenyl]-1,4-diazepane-1-carboxamide
1-methyl-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-({[(5-amino-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)-8-fluoroquinolin-4-ol
2-{4-[(6-chloropyridin-3-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetic acid
1-(2-methylpropyl)-8-(propan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N4,N4,5-trimethylpyrimidine-2,4-diamine
7-(2,6-dichlorobenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
4-(9H-fluorene-9-carbonyl)-1,4-oxazepan-6-ol
N-(1,1-dioxo-1λ6-thian-4-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-butyl-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
5-fluoro-N-[1-(1H-imidazol-1-yl)butan-2-yl]quinazolin-4-amine
N-cyclopropyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}pyridine-2-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amine
{1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-3-propylpiperidin-3-yl}methanol
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2,4-dimethoxyphenyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide