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ethyl 4-{3-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]propoxy}benzoate
methyl 4-{2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamido}butanoate
(1S,5R)-3-(5-amino-1H-pyrazole-3-carbonyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[(adamantan-2-yl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
(1R,5S,6R,7S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-3-(propan-2-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
prop-2-en-1-yl N-methyl-N-({1-[(3R,5S)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)carbamate
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylpropan-2-yl)acetamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4-(1H-pyrazol-1-yl)butan-1-one
1-[2-(3-methoxyphenyl)ethyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-[3-(5-methylfuran-2-yl)-5-[3-(pyrrolidin-1-yl)butyl]-1H-1,2,4-triazol-1-yl]acetic acid
1-phenyl-3-{2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl}urea
2-(2-methoxyethyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(carbamoylmethyl)piperidine-3-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-chloro-2-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
3-{[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]methyl}phenol
2-cyclopropyl-9-[4-(hydroxymethyl)cyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]sulfanyl}ethan-1-ol
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-(pyrrolidin-1-yl)acetamide
N-cyclopropyl-4-hydroxy-N-[(2-methoxyphenyl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-(1-methoxypropan-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-(1H-indol-5-ylmethyl)propanamide
N-cyclopropyl-3-(4-hydroxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-benzyl-3-ethyl-1-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-1,4-diazepan-5-one
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}acetic acid
9-[(2,4-dimethylphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
3-(pyrrolidine-1-carbonyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
3-(4-ethyl-1H-pyrazol-5-yl)-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine
({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl](quinoxalin-5-ylmethyl)amine
1-[2-(pent-4-enamido)ethyl]-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
3-[2-(2-fluorophenyl)ethyl]-1-(prop-2-ene-1-sulfonyl)piperidine
8-[(3-methylpyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
4-(5-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
methyl 6-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidine-4-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
(3S,7S)-5-(6-oxo-1,6-dihydropyridine-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(prop-2-en-1-yl)(propan-2-yl)amine
2-(4-{[(2-methoxyethyl)(methyl)amino]methyl}phenyl)-6-(3-methylpyrazin-2-yl)-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-(2,2-dimethylpropanoyl)-4-[(4-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexanecarbonyl-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
1-[3-(3-fluorophenyl)phenyl]-N-[1-(pyrimidin-4-yl)ethyl]piperidin-4-amine
4-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}thiomorpholine
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide