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1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
7-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-[3-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)phenoxy]acetamide
N-[4-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
3-(but-2-yn-1-yl)-5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrimidine-2,4-diamine
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)(pyridin-3-ylmethyl)amine
3-phenoxy-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(2S,4R)-4-amino-1-{[1-(2-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methyl}-N-ethylpyrrolidine-2-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(2-methoxyethyl)-1,2-oxazole-3-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-ethyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-3-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)ethyl]-4-pentanamidobenzamide
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-phenyl-1,2-oxazole-3-carboxamide
1-[(2,5-difluorophenyl)methyl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl][1-(5-methylpyridin-2-yl)propan-2-yl]amine
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(trifluoromethyl)pyridine
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
6-(dimethylamino)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyridine-3-carboxamide
{2-[(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}methanol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(methylsulfanyl)benzamide
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
1-[(4-chloro-3-fluorophenyl)methyl]-3-(1-ethyl-1H-imidazol-2-yl)piperidine
N1-phenyl-N2-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]ethane-1,2-diamine
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-4-[(propan-2-yl)sulfamoyl]benzamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(3-hydroxypropyl)-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2,2-dimethyloxan-4-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
(5-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-2-(propan-2-yloxy)phenyl)methanol
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}propanamide
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
methyl 2-{5-methyl-2-[(1,2,5-thiadiazol-3-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
methyl (2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
1-[(2-chlorophenyl)methyl]-5-[4-(2,3-dimethylphenyl)piperazin-1-yl]azepan-2-one
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-1-(naphthalen-2-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
[(3S,5R)-1-(2,6-dimethylpyrimidine-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenyl-N-(propan-2-yl)-1,2-oxazole-4-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
4-(6-methoxypyridin-2-yl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenol
2-(1-benzothiophen-3-yl)-5-methylpyrimidin-4-amine
4-[(2-hydroxyethyl)(methyl)amino]-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
8-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
7-(3-chlorophenyl)-9-methoxy-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4S)-4-amino-N-methyl-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
3-[5-({3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}methyl)thiophen-3-yl]prop-2-yn-1-ol
ethyl 3-benzyl-1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidine-3-carboxylate