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4-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]oxane-4-carbonitrile
1-(2-methanesulfonylethyl)-5-(pentan-2-yl)-4-phenyl-1H-imidazole
3-(2-methoxyphenoxy)-1-(2-phenylethyl)azetidine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
2-{4-methyl-6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-2-yl}phenol
1,5-dimethyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1H-pyrazole-4-carboxamide
2-{6-hydroxy-4-[(8-methoxy-2H-chromen-3-yl)methyl]-1,4-diazepan-1-yl}acetic acid
(2S,4R)-1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-methyl-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-methylpropanamide
8-(furan-2-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidine
1-(2-ethoxyethyl)-2-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]methylamine
dimethyl({4-methyl-5-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
(3aS,6aS)-1-methyl-N-(2-phenylethyl)-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(2S,4R)-4-amino-1-[3-(2-methoxyphenyl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
4-methyl-N-[phenyl(pyridin-4-yl)methyl]pyrimidine-5-carboxamide
4-(3-cyanopyridin-2-yl)-N-(2,3-dihydro-1H-inden-5-yl)piperazine-1-carboxamide
4-(4-chlorophenyl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}butan-1-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(1-methylpiperidin-4-yl)pyrimidin-2-amine
(3aR,6aR)-2-[2-(3-fluoro-4-methylphenyl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-methylphenoxy)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
3-(methanesulfonylmethyl)-N-[3-(3-methylphenyl)phenyl]piperidine-1-carboxamide
(2E)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
2-(benzyloxy)-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]acetamide
1-[4-(3-methylpiperidine-1-carbonyl)phenyl]-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethoxyethan-1-one
2-methoxy-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
4-methyl-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)pyrimidine-5-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
8-(3-ethyl-1H-pyrazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3S)-3-hydroxy-3-phenylpropyl]-4-(hydroxymethyl)piperidin-4-ol
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}butanamide
[2-({4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
1-(4-methoxyphenyl)-4-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}piperazine
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-3-carbonitrile
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
1-{5-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-5-carbonyl]thiophen-2-yl}ethan-1-one
4,4,4-trifluoro-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}butan-1-one