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1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-methyl-1,4-diazepan-5-one
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-carbamoylethyl)propanamide
4-(furan-2-ylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
9-ethyl-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-{[(butan-2-yl)(cyclopentyl)amino]methyl}benzonitrile
N-(1-carbamoylcyclopentyl)-3,6-dimethyl-1-benzofuran-2-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-methyl-N-(propan-2-yl)acetamide
4-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-7-fluoro-2-methylquinoline
4-(3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2,2-dimethylpropyl)morpholine
2-amino-4-(4-hydroxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
6-fluoro-4-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,2-dihydroquinolin-2-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methylpyrazine-2-carboxamide
1-{2-hydroxy-3-[4-methoxy-2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
5-methyl-5-(4-methylpent-3-en-1-yl)-1-(1,2-oxazol-3-ylmethyl)piperidin-2-one
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(propan-2-yl)pyridazine
2,5-dimethyl-3-{4-[(5-methylthiophen-2-yl)methyl]piperazin-1-yl}pyrazine
N-cyclobutyl-4-(2,6-difluorobenzenesulfonyl)morpholine-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(propane-1-sulfonyl)piperidin-3-yl]propanamide
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2-(propan-2-yl)pyrimidine
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
{4-propoxy-3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methanol
(3aR,6aR)-2-benzyl-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
N-methyl-3-{[2-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}benzamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-1,3-dimethyl-4-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(pyridin-2-yl)propanamide
1-cyclopentyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1,2-dihydroquinolin-2-one
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-8-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-[1-(4-methanesulfonylphenyl)-1H-imidazol-2-yl]pyridine
7-(cyclopropylmethyl)-2-[3-(dimethylamino)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(thiophen-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(4-{[3-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amine
4-(1H-imidazol-2-yl)-1-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1H-1,2,3-triazole
5-benzyl-4-(3-hydroxypropyl)-1-(3-phenylphenyl)piperazin-2-one
N-[2-(2-ethylphenoxy)ethyl]-N-methylquinoline-6-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(4aS,7aR)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[3-(1H-imidazol-1-yl)-1-phenylpropyl]carbamoyl}-1H-imidazole-4-carboxylic acid
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
4-(2-methyl-1H-imidazol-1-yl)-1-[(3-methylthiophen-2-yl)methyl]piperidine-4-carboxylic acid
2-[2-(azepan-1-ylmethyl)phenyl]-6-butyl-3,4-dihydropyrimidin-4-one
2-methyl-1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one