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N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-4-carboxamide
N-{1-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
N-[1-(2-phenylethyl)-7-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]methanesulfonamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(4-sulfamoylphenyl)ethyl]acetamide
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
2-fluoro-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
2-({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)-N,N-dimethylpropanamide
3-cyclohexyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-pyrazole-4-carboxamide
2-chloro-N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(4aS,8aR)-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
5-(2,6-difluorophenoxymethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2-oxazole-3-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-methyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
2-[1-methyl-4-(5-phenoxyfuran-2-carbonyl)piperazin-2-yl]ethan-1-ol
1-[2-(3-fluorophenyl)ethyl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[1-(2-fluorophenyl)-5-[2-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-methoxy-3-methylbenzene-1-sulfonamide
3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
(4aS,8aR)-6-(2-methoxyethyl)-1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,6-dimethylpyrimidin-2-amine
(1S,5R)-3-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1H-indol-3-yl)ethyl]-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea
(3R,4R)-1-(2-aminopyrimidin-4-yl)-4-(morpholin-4-yl)piperidin-3-ol
1-(piperazin-1-yl)-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
3-amino-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
N-(2-ethoxyethyl)-3-{[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]sulfonyl}benzamide
1,2-dimethyl-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1H-indol-5-ol
ethyl 2-(4-{[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]amino}phenyl)acetate
1-(carbamoylmethyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
3-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-5-phenyl-1,2,4-oxadiazole
(3aR,6aS)-2-{[2-(5-methylfuran-2-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole
4-(benzyloxy)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
(1R,9S)-5-amino-3-(2-fluoro-3-methoxyphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
3,5-dimethyl-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-(2,3,4-trimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
3-[2-(dimethylamino)ethyl]-8-(quinoline-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
[1-(1-methoxypropan-2-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
6,7-dimethoxy-3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydroquinazolin-4-one
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(prop-2-en-1-yl)amino]pyridine-3-carboxamide
1-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
6-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)pyridine-2-carbonitrile
N-ethyl-2-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]acetamide