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2-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}quinolin-4-ol
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
1-(2,3-dimethylphenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-cyclopentyl-N'-{[(1R,2R)-2-hydroxycyclohexyl]methyl}butanediamide
1-(3-methoxypropanoyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
1-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-fluorophenoxymethyl)-N-(pentan-3-yl)-1H-pyrazole-3-carboxamide
2-(4-phenylpiperidin-1-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
N-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-N,4-dimethyl-1,3-oxazole-5-carboxamide
2-({2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)-1,3-benzoxazole
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)[3-(oxolan-2-yl)propyl]amine
6-(2-chlorophenyl)-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
methyl 2-({3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)benzoate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(1S,4S)-5-(5,6-dimethylpyrimidin-4-yl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})methylamine
9-(3-hydroxybenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(1R,5R)-N-[(3-fluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[9-hydroxy-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
(2S,4S)-N-methyl-1-(1-propylpiperidin-4-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(3S,4R)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[2-(dimethylsulfamoyl)ethyl]-5,6-dimethylpyridine-3-carboxamide
2-[4-(2-methylpropyl)-1,4-diazepane-1-carbonyl]-N-(prop-2-en-1-yl)aniline
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-hydroxypropanoyl)piperidine-4-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-3-(1H-1,2,3-benzotriazol-1-yl)propanamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1,5-dimethyl-3-{[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indazole
1-benzyl-8-[(5-methylthiophen-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-6-[4-(2-methoxyethoxy)phenyl]-N-methylpyrimidin-4-amine
7-(4-chloro-1H-indole-2-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
2-(4-fluorophenoxymethyl)-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-1,3-oxazole-4-carboxamide
3-(1,4-diazepan-1-ylmethyl)-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-1-phenylpiperazin-2-one
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
(1R,9aR)-1-({[3-(pyridin-3-yloxy)propyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
8-[2-(2-oxopyrrolidin-1-yl)acetyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(quinolin-8-yl)-4-(thian-4-yl)piperazine-1-carboxamide
2-[2-(4-fluoro-3-methylbenzenesulfonamido)-N-methylacetamido]-N-methylpropanamide
3-{2-[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1'-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N,N-dimethyl-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
1-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidine-4-carboxamide