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ethyl 4-{7-chloro-3-[(N-cyclopropyl-1-1,3-thiazol-5-ylformamido)methyl]quinolin-2-yl}piperazine-1-carboxylate
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-ethoxyethan-1-one
(2R,3R)-3-(dimethylamino)-1'-(2-methylfuran-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-diethylpyrrolidin-3-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]benzamide
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(1H-indol-4-ylmethyl)acetamide
N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-(4-fluorophenyl)-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]cyclopropane-1-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]propanamide
5-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
4-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]-N-(propan-2-yl)pyridine-2-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[2-(4-ethylphenoxy)ethyl]-N-methylpent-4-ynamide
1-(furan-2-ylmethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
5-methoxy-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4-oxo-1,4-dihydropyridine-2-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
2-methyl-4-(5-{1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)but-3-yn-2-ol
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4S)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
6-{5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazol-1-yl}-2-methyl-1,3-benzothiazole
3-(1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)propan-1-ol
N-(3-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-oxopropyl)-N-methylmethanesulfonamide
2-methyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(propan-2-yl)pyrimidine
1-(cyclopent-1-ene-1-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-3-carboxamide
methyl 2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}benzoate
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-{1-[(2-chlorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
2-hydroxy-5-methoxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
methyl 3-(1-phenylcyclopropaneamido)-6-(thiomorpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
1-(4-chlorophenyl)-N-{[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
3-[5-(7-fluoro-4-methylquinolin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
5-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-1,3-benzothiazole
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}propanamide
7-[(3,4-difluorophenyl)methyl]-2-propanoyl-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-fluorophenyl)ethyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
4-methyl-2-{1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}-3,4-dihydro-2H-1,4-benzoxazine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(5-ethylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3R,4S)-1-[(4-chloro-3-fluorophenyl)methyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
5-[3-(1-butyl-1H-pyrazol-3-yl)phenyl]pyrimidine
2-(adamantan-1-yl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpent-3-en-1-yl)piperidine
4-{4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]piperidin-1-yl}-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}thiolan-3-amine
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine