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4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-phenylurea
4-acetyl-1-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-2-one
1-[1-(1,2-oxazole-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(5-oxopyrrolidin-2-yl)acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2-methyl-1H-indol-3-yl)acetamide
N-(4-chloro-3-fluorophenyl)-4-(2-methylpyrimidin-4-yl)piperidine-1-carboxamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(3-methoxypiperidin-1-yl)pyridine
(1-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}piperidin-3-yl)methanol
5-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-(azepane-1-carbonyl)-N-[(1-hydroxycyclohexyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
5-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
methyl 4-{5-[(3-propoxypiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{[6-(4-methanesulfonylphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
N-(2-hydroxyethyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(4aS,8aR)-6-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
5-ethyl-2-methyl-4-[4-(2,2,6,6-tetramethylpiperidin-4-yl)piperazin-1-yl]pyrimidine
[(4-methoxyphenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-methyl-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)propan-1-ol
(3R,4S)-4-cyclopropyl-1-(3-fluorobenzenesulfonyl)pyrrolidin-3-amine
1'-[4-(4H-1,2,4-triazol-4-yl)benzoyl]spiro[indene-1,4'-piperidine]
(3R,4R)-1-{[4-(difluoromethoxy)phenyl]methyl}-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
ethyl 4-(2,6-dimethoxyphenyl)-2-(methylsulfanyl)pyrimidine-5-carboxylate
N-(3-hydroxy-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)acetamide
(1S,6R)-3-methyl-9-[(5-methylthiophen-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
ethyl 5-(1H-imidazol-2-ylmethyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2-hydroxyethyl)-8-[2-(1H-indol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methylphenyl)-2-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]acetamide
4-methyl-2-(pyridin-3-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
2-(prop-2-en-1-yl)-4-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)phenol
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
[4-({methyl[(2E)-4-methylpent-2-en-1-yl]amino}methyl)oxan-4-yl]methanol
2-[4-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
4-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]benzoic acid
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-2-one
2-(4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperazin-1-yl)pyrimidine
3-methoxy-1-[2-(1-methylpiperidin-2-yl)ethyl]-1,2-dihydropyridin-2-one
5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-benzotriazole
3-[(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
1-(oxane-4-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide