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methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(2-methylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[7-(pyridin-3-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}cyclopent-1-ene-1-carboxamide
2-{1-cyclopentyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-amino-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-ethylphenyl)methyl]-N-[(2-methoxyphenyl)methyl]-2-(morpholin-3-yl)acetamide
4-ethyl-N,N-dimethyl-6-{4-[methyl(oxan-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-amine
3,5-dimethoxy-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2,3-dimethoxy-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]benzamide
(4aS,8aR)-1-(3-aminopropyl)-6-(2-methyl-6-propylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
1-{4-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]thiophen-2-yl}ethan-1-one
3-chloro-N-cyclopentyl-4-{[1-(pyridine-4-carbonyl)piperidin-4-yl]oxy}benzamide
1-(3-chlorophenyl)-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methylpiperazin-2-one
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
8-[2-(azepan-1-yl)-2-oxoethyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-7-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]but-2-yn-1-one
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-(3-fluorophenyl)-3-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
7-methoxy-3-(1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(1,3-thiazol-4-ylmethyl)piperidine
1,3-dimethyl-6-(pyridin-4-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-acetylphenoxy)-1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
8-(2,3-dihydro-1H-indene-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1'-{[4-(prop-2-en-1-yloxy)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]benzoic acid
N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
methyl 3-(4-methoxybenzamido)-1-methyl-5-{[1-(methylsulfanyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2,3,5,6-tetramethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)benzamide
methyl 4-(2-benzyl-3-oxopiperazine-1-carbonyl)benzoate
N-methyl-N-(propan-2-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-1-phenylpiperazin-2-one
5-(piperidin-1-ylmethyl)-2-(1H-pyrazol-4-yl)pyridine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-(1H-pyrazol-1-yl)acetamide
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-4-{3-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
2-{3-[3-(6-methylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-(2-hydroxy-2-methylpropanoyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
ethyl 3-benzyl-1-[(5-acetamidoquinolin-2-yl)methyl]piperidine-3-carboxylate
1-(2-ethoxyphenyl)-4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazine
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-{1-[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
{1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N-[2-fluoro-5-(trifluoromethyl)phenyl]-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carboxamide
2-[(5-fluoro-2-methylphenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide