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5-[2-(4-fluorophenyl)morpholine-4-carbonyl]-4-phenylpyrimidin-2-amine
2-(methylsulfanyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3-thiazole-4-carboxamide
2-ethyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyrimidine-5-carboxamide
2-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1'-[6-(morpholin-4-yl)pyrimidin-4-yl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol
N-(2-methyl-1,3-benzothiazol-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrrol-1-yl)propan-1-one
1-[(2,4-dimethylphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(4-fluorophenyl)methyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}propanamide
1-(4-fluorophenyl)-4-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}butane-1,4-dione
[1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-(furan-2-ylmethyl)-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine-2-carboxamide
2-(1-benzyl-4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-(furan-2-ylmethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
5-cyclobutanecarbonyl-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{4-[1-(dimethylamino)ethyl]phenyl}benzonitrile
N-[3-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
2-(2,3-dimethoxyphenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
1-[4-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-chloro-2-propanamido-N-[(1-propylpiperidin-4-yl)methyl]benzamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-chloro-1,2-dihydropyridin-2-one
2-[(3-methoxyphenyl)methyl]-8-(4-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
dimethyl(1-{4-[1-(quinoxalin-6-yl)-1H-imidazol-2-yl]phenyl}ethyl)amine
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-methylbutan-1-one
3-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2,3,6-trifluorophenyl)acetamide
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2-(2,3,6-trimethylphenoxy)acetamide
1-{[1-(2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}acetyl)piperidin-3-yl]methyl}pyrrolidin-2-one
1-(cyclopropylmethyl)-4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-2-(propan-2-yl)-1,4-diazepane
4-[(6-chloro-2H-chromen-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methyl-1-[3-(piperidin-1-ylmethyl)phenyl]urea
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-(furan-2-ylmethyl)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]-N-(2-phenylethyl)benzamide
N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-methoxy-N-methylbenzamide
N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-methyl-8-[2-(pyridin-2-yl)pyrimidin-5-yl]-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
methyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-[(3,4-difluorophenyl)methyl]-3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-[(2,3-difluorophenyl)methyl]-4-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]piperidine
6-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methoxyhexan-1-one
7-cyclopentyl-2-(2-methanesulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-(2-hydroxyethyl)-3-[5-(thiophen-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
methyl 6-(pent-4-enoyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate