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6-cyclopentyl-1-methyl-N-[5-(morpholin-4-yl)pentyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(3-methoxyphenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
methyl 5-(5-methoxyfuran-2-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
1-cyclohexyl-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-N'-(2-methylphenyl)propanediamide
8-(2,3-dihydro-1H-indene-1-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
4-(2,6-dimethylpyridin-3-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrimidin-2-amine
[(1-cyclopentylpiperidin-4-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
7-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-ethanesulfonamido-1-methyl-N-(oxolan-2-ylmethyl)-2-phenyl-N-propyl-1H-1,3-benzodiazole-7-carboxamide
5-(2,5-dimethylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidine
4-[1-(4-fluorophenyl)propan-2-yl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-({1-[6-(azepan-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-{4-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-(2,5-dimethoxyphenyl)acetic acid
5-(methoxymethyl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
2-(3-fluorophenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-N-(prop-2-en-1-yl)piperidine-1-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(methylsulfanyl)pyrimidin-4-yl]-1-(pyrrolidine-1-carbonyl)azepan-3-amine
2-[2-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)phenoxy]acetamide
5-{[(4-fluorophenyl)methyl]amino}-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}benzoic acid
4-({2-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
2-(adamantan-1-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-hydroxypyrimidine-5-carboxamide
N2-[6-(propan-2-yl)pyrimidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(benzenesulfonyl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
ethyl 1,5-bis(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[4-(4-oxo-4H-chromen-7-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(cyclohexylmethyl)-N-ethyl-3-(3-hydroxy-3-methylbutyl)benzamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1H-imidazol-1-yl)butan-2-yl]-1,3-oxazole-4-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide
3-cyclohexyl-N-[2-(1H-imidazol-4-yl)ethyl]-1H-pyrazole-4-carboxamide
7-methyl-2-[2-(3-oxopiperazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
6-(2-chlorophenyl)-N-(2,2-difluoroethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-methoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
5-(3-methoxyphenyl)-2-(pyridin-4-yl)-4-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]pyrimidine
3-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
4-{[benzyl(methyl)amino]methyl}-1-cyclopentylpyrrolidin-2-one
[(2-ethylpyrimidin-4-yl)methyl][2-(1H-indol-1-yl)ethyl]methylamine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-1-(1,3-thiazol-4-ylmethyl)piperidine