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3-(2-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxyphenyl)propanamide
(2-methoxyethyl)[(4-methoxyphenyl)methyl]({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
3-(4-methoxyphenoxymethyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
(4aS,8aS)-2-[4-(4-methylpiperazin-1-yl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
(2S,4R)-4-amino-N-methyl-1-{3-[(4-methylphenyl)formamido]propanoyl}pyrrolidine-2-carboxamide
2-(3-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}piperidin-1-yl)acetamide
2-{4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
4-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
2-chloro-N-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[3-(3-chlorophenyl)phenyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxamide
N-[2-(2-phenoxyethoxy)phenyl]-1H-pyrazole-3-carboxamide
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N,N-dimethylpropane-1-sulfonamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-{1'-[(2,4-difluorophenyl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
N-(1-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
methyl 4-[4-({1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
(3aS,6aS)-2-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(1H-imidazol-1-yl)propyl]-8-methyl-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
9-methoxy-7-(3-methoxyphenyl)-4-(1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-fluorophenyl)-N-[(3-methyloxetan-3-yl)methyl]benzamide
2,5-dimethyl-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}-3-methylbenzamide
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{3-[(3-hydroxy-3-phenylpyrrolidin-1-yl)methyl]phenyl}-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,6-dimethyl-N-(pyridin-4-ylmethyl)pyrimidine-4-carboxamide
(2S,4S)-4-(3,5-difluorobenzamido)-N-(3-methoxypropyl)-1-methylpyrrolidine-2-carboxamide
3-[5-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
7-(2-methoxyethyl)-2-{thieno[3,2-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
N-(2-acetylphenyl)-3-{[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}propanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-methoxy-2-methylpropanamide
4'-[1-(azepan-1-yl)-1-oxopropan-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-chloro-4-fluorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]furan-3-carboxamide
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}benzamide
4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)benzoic acid
1-{4-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{3-[1-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]propyl}piperidin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(4-sulfamoylbenzoyl)piperidin-3-yl]propanoic acid
2-(2-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
2-(4-benzylmorpholin-2-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(2-methylpropyl)acetamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)acetamide
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1,4-diazepane-1-carboxamide