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2-[3-(2,4-dimethylphenyl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
3-(4-methoxyphenyl)-N-methyl-N-(2-methylprop-2-en-1-yl)-3-phenylpropanamide
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-amino-6-benzoyl-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-butyl-N-(3-chloro-4-fluorophenyl)-4-methyl-3-oxopiperazine-1-carboxamide
3-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}pyridine
1-cyclopropyl-5-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-2-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[3-(methylsulfanyl)propyl]piperidin-4-ol
[(1-benzylpyrrolidin-3-yl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-(2,3-dihydroxypropyl)-6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylpiperidin-4-yl)piperidine
2-{4-methyl-6-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidin-2-yl}phenol
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(4-fluorophenyl)ethyl]propanamide
(3S,4S)-4-(morpholin-4-yl)-1-(pyrimidin-2-yl)pyrrolidin-3-ol
2,3-dimethoxy-N-{[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}benzamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-amine
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
1-(6-hydroxy-4-{[2-(propylamino)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}acetamide
6-(4-fluorophenyl)-7-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-hydroxyphenyl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-methoxypropan-1-one
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
ethyl 6-methyl-2-(4-phenylazepan-1-yl)pyrimidine-4-carboxylate
1-(2-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-oxoethyl)-3-butyl-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 5-{[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-(pyridin-2-yl)-1H-pyrazole-4-carboxylate
2-methyl-5-[4-(piperidine-1-sulfonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
4-(3-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}propoxy)benzamide
(2S)-2-amino-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-benzyl-5-{[(3-fluorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl N-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)carbamate
3-(4-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}phenyl)prop-2-yn-1-ol
4-(2-methoxyphenoxy)-1-(pyridine-4-carbonyl)piperidine-4-carboxylic acid
N-(3-methoxypropyl)-1-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-amine
N-[(4-fluorophenyl)methyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
N,5-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{2-[(4-methoxy-4-methylpentan-2-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
4-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
2-hydroxy-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
3-({[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
3-methoxy-5-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}thiophene-2-carboxamide
7-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(cyclopropylmethyl)-1-(1,3-thiazol-2-yl)piperidine-3-carboxylic acid
3-[4-(5-chloro-2-methoxypyridin-4-yl)-1H-pyrazol-1-yl]propanamide
[(2S,6S)-4-[(3,5-dichloropyridin-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-({1-[2-(carbamoylamino)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-4-methylbenzamide