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2-{[4-(3-chlorophenyl)-5-[hydroxy(phenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(dimethylamino)-N-(1-{7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
ethyl 4-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)-1H-pyrazole-3-carboxylate
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methylpiperidine
2-(1-benzyl-4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
(4aS,7aR)-1-[(5-ethylpyridin-2-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-methylphenoxy)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxamide
5-[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile
1-[4-(pyrimidin-2-yl)piperazin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-ethyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrrolidin-2-one
3-(1H-indazol-7-yl)-1-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]urea
6-[(3-fluorophenyl)methoxy]-4-(1H-imidazole-4-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
4-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-4-oxobutanamide
N-ethyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophene-2-carboxamide
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,2-oxazole-3-carbonyl)piperidin-3-yl]methanol
4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-oxazepane
N-cyclopropyl-3-(3-hydroxy-3-methylbutyl)-N-propylbenzamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-methoxypropanamide
(3R,9R)-N-cyclohexyl-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxamide
N-(3-butoxyphenyl)-2-(2-hydroxyethyl)pyrrolidine-1-carboxamide
8-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-methoxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(3aR,5S,6S,7aS)-2-(2,6-difluoro-3-methylbenzoyl)-octahydro-1H-isoindole-5,6-diol
3-phenyl-3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-ol
2-cyclopropyl-9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
6-fluoro-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[(3-{[2-(2-aminoethyl)quinazolin-4-yl]amino}propyl)(2-hydroxyethyl)amino]ethan-1-ol
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]pyridin-2-amine
4-(4-fluorophenyl)-5-methyl-2-[5-(propan-2-yl)-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]pyrimidine
N,3,5-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-4-carboxamide
1-(4-{2-[3-(3-hydroxypropyl)piperidine-1-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-3-carbonyl]pyridine
N-cyclopropyl-3-({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}sulfamoyl)benzamide
N-tert-butyl-2-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]benzene-1-sulfonamide
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
8-[(3-chloro-4,5-dimethoxyphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[(1-{2-[ethyl(methyl)amino]acetyl}piperidin-4-yl)methyl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-methyl-N-(pentan-3-yl)-N-(2-phenylethyl)-1H-imidazole-5-carboxamide
7-(2-methoxyethyl)-2-(4-phenylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclohexyl-3-(cyclopropylmethyl)-N-[2-(1H-imidazol-1-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-ethanesulfonamido-1-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
(2R,3R,6R)-3-phenyl-5-(3-propyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-ethyl-N-[2-(1H-indol-1-yl)ethyl]-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[(3S,5S)-5-{[(1-hydroxycyclohexyl)methyl]carbamoyl}-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-(9-{[4-(methylsulfanyl)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide