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9-[2-(4-hydroxyphenyl)acetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-chloro-3-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
{2,2-dimethyl-3-[4-(5-methyl-1,3,4-thiadiazol-2-yl)piperazin-1-yl]propyl}dimethylamine
1-{2-[1-(4-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3,3,3-trifluoropropan-1-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
2,5-dimethyl-3-[4-(pyridin-4-ylmethyl)piperazin-1-yl]pyrazine
N-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
(3R,4S)-1-(2,6-dimethylpyridine-4-carbonyl)-4-propylpyrrolidin-3-amine
3-(3-chlorobenzoyl)-1-(2-chlorobenzenesulfonyl)piperidine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-(piperidin-4-ylmethyl)benzamide
4-(3,5-dimethyl-1H-indole-2-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
1-[4-(pyrrolidin-1-yl)benzoyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
8-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
6-fluoro-2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}quinolin-4-ol
[1-(azepan-1-yl)propan-2-yl][(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-(1-phenylpiperidin-4-yl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
5-chloro-N-[(4-methyl-1H-imidazol-2-yl)methyl]thiophene-2-carboxamide
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-{[5-fluoro-2-(1-methyl-1H-pyrazol-4-yl)pyrimidin-4-yl]amino}ethan-1-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
6-[3-(dimethylamino)phenyl]-N,N-dimethylpyridine-3-carboxamide
3-(hydroxymethyl)-N-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)piperidine-1-carboxamide
3-methoxy-1-{[4-(3-methylphenyl)phenyl]methyl}pyrrolidine
2-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-4,6-dimethylpyridine-3-carbonitrile
3-{3-[(4-propylpiperazin-1-yl)methyl]-1H-indol-1-yl}propanamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-methoxyfuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-hydroxyethyl)-2-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{[1-(3-methanesulfonylpropanoyl)pyrrolidin-3-yl]methyl}benzamide
N'-(2,4-dimethylphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanediamide
methyl[(1-phenylpyrrolidin-3-yl)methyl](1,3-thiazol-4-ylmethyl)amine
1-[(3-methylpyrazin-2-yl)methyl]-3-propylpiperidine-3-carboxylic acid
3,3-dimethyl-1-{2-[(3-methylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}butan-1-one
2-(3-fluorophenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-methyl-1-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]azetidin-3-yl}piperidine
1-(1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1,3-thiazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
(2S)-1-{2-[(2-methylphenyl)carbamoyl]acetyl}pyrrolidine-2-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
(3aS,6aS)-2-(3-methoxybenzoyl)-5-[3-(methylsulfanyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(naphthalen-1-ylmethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
6-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
2-[({5-[1-(2,6-diaminopyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide