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1'-(1-methyl-1H-pyrazole-5-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-ethoxy-4-{5-[(4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
5-phenyl-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
3-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
6-tert-butyl-2-oxo-N-(1-propylpyrrolidin-3-yl)-2,3-dihydropyrimidine-4-carboxamide
[(2S,6S)-4-[2-(4-fluorophenoxy)ethyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)methyl]-1-methyl-1,2-dihydroquinolin-2-one
(1R,5R)-3-benzoyl-6-(pent-2-yn-1-yl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aS)-2-(ethanesulfonyl)-5-[2-(pyridin-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3-methoxyphenyl)methyl]-4-(thiophene-3-sulfonyl)morpholine
7-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
1-[(4,6-dimethylpyridin-2-yl)methyl]-3-(5-methanesulfonamido-2-methylphenyl)-1-methylurea
5-{1-[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
1-{2-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}pyrrolidin-2-one
3-(4-hydroxyphenyl)-N-[2-(propylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
3-(3-cyano-4-methoxyphenyl)-1-[1-(cyclohex-1-en-1-yl)ethyl]urea
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-benzyl-decahydro-1,6-naphthyridin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[2-amino-4-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
9-[2-(6-methylpyridin-2-yl)ethyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(1-ethylpiperidin-4-yl)piperidine
N-{[1-(propan-2-yl)cyclopropyl]methyl}-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-ethyl-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(3,5-difluorobenzoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
4-ethyl-1-methyl-3-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-hydroxyethyl)-1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
7-(2-hydroxyethyl)-2-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]benzoate
methyl({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})(pyrimidin-4-ylmethyl)amine
N-(2-hydroxy-2-phenylethyl)-N-methyl-3-(quinolin-8-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[(3S,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
8-[6-(hydroxymethyl)pyridine-2-carbonyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(dimethylamino)butyl]-1,3-oxazole-4-carboxamide
N-(oxolan-2-ylmethyl)-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-benzyl-2-(morpholin-2-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
4-(1-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}azetidin-3-yl)morpholine
N,N-dimethyl-2-[(1S,5R)-3-(naphthalene-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-[(2,5-difluorophenyl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(4-amino-6,7-dimethoxyquinazolin-2-yl)benzonitrile
8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
(4S)-N-(2,4-dichlorophenyl)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide