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1-[2-(dimethylamino)ethyl]-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}pyridine
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-N-propylpyrimidin-2-amine
2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(1R,3S,5S)-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-8-azabicyclo[3.2.1]octan-3-ol
2-methyl-4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]phenol
(3R,4R)-1-(2-methoxy-4-methylbenzenesulfonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(3S)-N,N-dimethyl-1-[1-(4-methylphenyl)piperidin-4-yl]azepan-3-amine
(4aS,7aR)-1-(5-hydroxypyrazine-2-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
4-{[1-(cyclohexylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
9-benzyl-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-[2-(benzyloxy)ethyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
4-(6-methylhept-5-en-2-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-(benzyloxy)-1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidine
(2S,4S)-4-amino-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-methylpyrrolidine-2-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(1-ethylpiperidin-3-yl)piperidine
3-(2,6-dimethylphenoxy)-N-[3-(2-methoxyethoxy)phenyl]azetidine-1-carboxamide
3-(2-oxopyrrolidin-1-yl)-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-4-yl)pyrrolidin-3-yl]propanamide
4-{[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-propylpyrrolidin-1-yl]methyl}benzonitrile
[(2,4-difluorophenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-[4-methyl-6-(4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-yl]phenol
2-(3-cyclopropyl-5-{[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-1-yl)pyridine
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[2-(quinolin-3-yl)pyrimidin-4-yl]pyrrolidin-3-ol
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(4-phenoxybenzoyl)piperidine
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-3-(2-oxooxolan-3-yl)propanamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-2-methylpiperidine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-5-phenylpentanamide
2-methoxy-4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethan-1-ol
1-methyl-4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-(phenylsulfanyl)propyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-3,4-dimethoxypyridine
N-({7-[4-(4-methylphenyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
(3S,4S)-1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
ethyl 5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(3-methylbut-2-en-1-yl)-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl]ethan-1-ol
(4aS,8aR)-6-(3,5-difluoropyridine-2-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one