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2-(3-methoxypropyl)-9-phenylmethanesulfonyl-2,9-diazaspiro[5.5]undecan-3-one
1-({4-[3-(benzyloxy)azetidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
N-cyclopropyl-4-methoxy-3-({1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
N-(butan-2-yl)-N-[(2-chlorophenyl)methyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N-[(4-chlorophenyl)methyl]-N-cyclopropyl-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
7-methanesulfonyl-4-methyl-2-[2-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrrolidin-1-yl]quinazoline
6-(cyclopentylamino)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[1-(6-methylpyridin-3-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
4-{3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
{3-[(2,4-difluorophenyl)methyl]-1-(quinolin-2-yl)piperidin-3-yl}methanol
1-methyl-8-[3-(methylsulfanyl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(4aS,8aS)-N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-4a-hydroxy-decahydroisoquinoline-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(methylamino)acetyl]piperazin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-(pyrrolidin-1-yl)ethan-1-one
5-[6-(azepan-1-yl)pyridazin-3-yl]-1,2,3,4-tetrahydroisoquinoline
methyl 3-(furan-2-amido)-5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(5S,9aS,9bS)-5-(6-methoxy-2H-chromen-3-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
2-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]pyridine-3-carboxylic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)ethane-1-sulfonamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
(3S,4S)-4-(dimethylamino)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-ol
[1-(2-methyl-1,3-thiazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-methyl-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
3-oxo-N-(2-phenoxyphenyl)-2,8-diazaspiro[4.5]decane-8-carboxamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)pent-4-enamide
(3R,4S)-3,4-dimethyl-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
9-hydroxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
[(3R,4R)-1-(3-methyl-1-benzothiophene-2-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N,N-dimethyl-7-(5-methylpyridine-3-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-N,N-dimethylpyrimidin-2-amine
1-[(3-methylphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(pyrrolidin-1-yl)butan-1-one
4,5,6-trimethyl-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-ethyl-N,2-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrimidin-4-amine
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)amine
4-(1H-imidazol-1-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}benzamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-methoxypyrimidin-4-amine
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
(1R,3S)-7-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]acetamide
1-amino-N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]cyclopropane-1-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methylpyridine
1-{[3-methoxy-4-(4-methoxy-3-methylphenoxy)phenyl]methyl}pyrrolidine
N-{[3-methyl-7-(thiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide