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2,7-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]imidazo[1,2-a]pyridine-3-carboxamide
(3R,4R)-3,4-dimethyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-ol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-hydroxypropanoyl)pyrrolidine-3-carboxylic acid
5,8-dimethoxy-N,4-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]quinolin-2-amine
2-[(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)oxy]pyrimidine
N-(2-phenylethyl)-1-{2-[(pyridin-3-ylmethyl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-chloro-5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
2-(cyclopropylmethyl)-8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]butanoate
5-ethyl-6-methyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-(pyridin-4-ylsulfanyl)-N-[1-(thiophen-2-yl)ethyl]acetamide
N-methyl-3-(2-methyl-1H-imidazol-1-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
7-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-oxa-7-azaspiro[3.5]nonane
(3S)-3-({5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
3-(3-chlorophenyl)-1-(cyclopropylmethyl)-6-(1,2-oxazole-5-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(2-{[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
2,5-dimethyl-3-[4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]pyrazine
9-(1H-indol-3-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-(3-methylbut-2-en-1-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
(4aS,7aR)-1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 2-{[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}-2-methylpropanoate
(1r,4r)-4-[({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]cyclohexan-1-ol
3,5-dimethyl-N-[1-(pyridin-4-yl)propyl]-1-benzofuran-2-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3,4-dimethoxybenzoyl)piperidine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-ethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(thiophen-3-ylmethyl)acetamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
N-(2-methoxyethyl)-1-{1-[6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
(2S,3R)-2-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-hydroxybutanamide
N-(2-methoxyethyl)-2-(methylamino)-N-(naphthalen-1-ylmethyl)pyrimidine-5-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(2,2,2-trifluoroethyl)acetamide
2-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(cyclobutylmethyl)-3-methyl-N-(oxolan-2-ylmethyl)but-2-enamide
6-cyclopentyl-1-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-chloro-6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyridazine
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
(3S,4S)-1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethylpyrimidine-5-carboxamide
(4S,4aS,8aS)-1-[(3-hydroxyphenyl)methyl]-4-phenyl-decahydroquinolin-4-ol
(2S,4S)-4-amino-N-ethyl-1-[(2S)-2-(6-methoxynaphthalen-2-yl)propanoyl]pyrrolidine-2-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-4-methyl-1H-pyrazole-5-carboxamide
4-(2-methoxyethyl)-1-(4-phenylbutan-2-yl)-1,4-diazepan-5-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-amine
2-[(4-chlorophenyl)methyl]-N-(oxan-4-ylmethyl)benzamide
3-[(3R,4S)-3-[2-(2-oxoazepan-1-yl)acetamido]-4-propylpyrrolidin-1-yl]propanamide