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N,N-dimethyl-2-{[2-(3-methylphenyl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}piperidin-2-one
(2S,4R)-4-amino-1-[(2S)-2-(6-methoxynaphthalen-2-yl)propanoyl]-N-methylpyrrolidine-2-carboxamide
[9-(1H-imidazol-4-ylmethyl)-3-(5-methoxyfuran-2-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-ethoxypropan-1-one
4-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-2-carboxylic acid
3-{[1-(furan-2-carbonyl)piperidin-4-yl]amino}-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
2,3,5-trimethyl-7-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}pyrazolo[1,5-a]pyrimidine
4-hydroxy-N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
1-methyl-6-(propan-2-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6,7-difluoro-3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-methylacetamide
3-(4-methylphenoxy)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)azetidine
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
ethyl 5-{[4-(2,5-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
2-ethyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrimidine
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-{4-[(5-cyclohexylthiophen-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[(1S,5R)-6-(5-ethylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[(dimethylamino)methyl]-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-[4-(2-ethylpiperidine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
2-(3,4-dichlorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-cyclohexyl-3-cyclopentyl-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
(3E)-5,5-dimethyl-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]hex-3-enoic acid
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl}acetamide
2-(cyclohex-1-en-1-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(3S,5R)-1-[(3-methoxyphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(4-fluorophenyl)-N-(2,2,2-trifluoroethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(4-chlorophenyl)ethyl]-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}propyl)-N-methyl-1H-1,2,3-triazole-5-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
1-[4-(3-methoxypiperidin-1-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(2-fluoroethyl)-3-{[4-(morpholin-4-yl)butan-2-yl]sulfamoyl}benzamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
4-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-2-(2-phenylethyl)morpholine
(2R,3R)-3-amino-1'-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(2-hydroxyphenyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]-1H-pyrazole-5-carboxamide
3-{5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanamide