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N-[2-(dimethylamino)ethyl]-4-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][(4-phenyl-1,3-thiazol-2-yl)methyl]amine
2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-(piperidin-4-yl)pyridine-3-carbonitrile
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
3-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,9-diazaspiro[5.5]undecane
1-{2-oxo-2-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyridin-2-one
3-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[1-(6-ethyl-2-methylquinoline-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
2-(cycloheptylamino)-N-(propan-2-yl)acetamide
2-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
2-methyl-4-phenyl-9-(thiophen-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2,7-diazaspiro[4.5]decane-7-carbonyl}-4-(1H-pyrrol-1-yl)phenol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}piperazine
(1S,5R)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
9-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-(2-methoxy-4-{[(3-methoxypropyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}piperidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methoxybenzenesulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2,3-dimethoxyphenyl)methyl]-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane
1-(oxolan-2-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(thiophene-2-carbonyl)piperazine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
ethyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
5-methoxy-9-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-(1,4-dioxan-2-ylmethyl)-1-benzofuran-2-carboxamide
(3R,5S)-N-(3-phenoxypropyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
4-(1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methoxyphenol
6-(2,3-dimethoxyphenyl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
4-{[1-(2-methanesulfonamidoacetyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(azocan-1-yl)-2-(5-fluoro-2-methoxyphenyl)acetic acid
2-(2,5-dimethylphenyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-(4-{1-[(2-methylpyridin-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)acetamide
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
2-(3-fluorophenoxy)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
4-phenyl-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidin-2-amine
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methoxy-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
(4aR,7aS)-1-methanesulfonyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,9S)-5-amino-3-(3-ethyl-1,2-oxazol-5-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
3-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)carbamoyl}amino)-N,4-dimethylbenzamide
N,N-dimethyl-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-sulfonamide